SCHEMBL6374657

SCHEMBL6374657

CCCC(NC(=O)Nc1ccccc1)C(=O)NCc1ccccc1-c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
FPR2 P25090 4/20 0.48
KCNA5 P22460 1/20 0.47
TAS1R3 Q7RTX0 1/20 0.44
TAS1R1 Q7RTX1 1/20 0.44
TSHR P16473 2/20 0.42
MAPT P10636 1/20 0.41
PSMB5 P28074 1/20 0.41
EPHX1 P07099 3/20 0.40
ALDH1A1 P00352 1/20 0.40
HTT P42858 1/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
MME P08473 1/20 0.40
ACE P12821 1/20 0.40
CPA1 P15085 1/20 0.40
ACE2 Q9BYF1 1/20 0.40
HSD17B10 Q99714 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6373116 0.85 FPR2 (0.51) MEN1KMT2AFPR2ALDH1A1
SCHEMBL6376129 0.85 FPR2 (0.51) MEN1KMT2AFPR2ALDH1A1
SCHEMBL6373106 0.85 FPR2 (0.51) MEN1KMT2AFPR2ALDH1A1
SCHEMBL6376146 0.80 RORC (0.47) MEN1KMT2AFPR2NPC1RAB9A
SCHEMBL6374484 0.77 FPR2 (0.76) KMT2AFPR2TSHRMAPTEPHX1
SCHEMBL6379257 0.77 FPR2 (0.76) KMT2AFPR2TSHRMAPTEPHX1
SCHEMBL6374491 0.77 FPR2 (0.76) KMT2AFPR2TSHRMAPTEPHX1
SCHEMBL6375041 0.76 FPR2 (0.47) MEN1KMT2AFPR2MAPTALDH1A1
SCHEMBL6376658 0.76 FPR2 (0.47) MEN1KMT2AFPR2MAPTALDH1A1
SCHEMBL15831236 0.75 KMT2A (0.53) MEN1KMT2AKCNA5ALDH1A1MME

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050137230-A1 Carboxamide derivatives DORSCH DIETER (DE) 2005-06-23 US claimed
US-20040038858-A1 Carboxamide derivatives and their use in the treatment of thromboembolic diseases and tumours MERCK PATENT GMBH (DE) 2004-02-26 US claimed
US-20050137230-A1 Carboxamide derivatives DORSCH DIETER (DE) 2005-06-23 US disclosed
US-20040038858-A1 Carboxamide derivatives and their use in the treatment of thromboembolic diseases and tumours MERCK PATENT GMBH (DE) 2004-02-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050137230-A1 Carboxamide derivatives F11, F12, F2 MEN1 218/4885KMT2A 1277/4885FPR2 766/4885
US-20040038858-A1 Carboxamide derivatives and their use in the treatment of thromboembolic diseases and tumours CNR2, CNR1, HCAR2 MEN1 3354/4885KMT2A 697/4885FPR2 176/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.