SCHEMBL6375219

SCHEMBL6375219

COc1cc(C(OC(C)=O)c2ccccc2)ccn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
CYP3A4 P08684 1/20 0.40
KMT2A Q03164 2/20 0.39
PABPC1 P11940 1/20 0.39
APOBEC3A P31941 1/20 0.39
APOBEC3G Q9HC16 1/20 0.39
POLB P06746 1/20 0.39
CTSA P10619 1/20 0.38
NCOA3 Q9Y6Q9 1/20 0.38
HSD17B10 Q99714 1/20 0.38
IDO1 P14902 1/20 0.38
MAPK1 P28482 1/20 0.37
ROCK2 O75116 1/20 0.37
ESR1 P03372 1/20 0.37
ESR2 Q92731 1/20 0.37
FFAR1 O14842 1/20 0.36
HTR1A P08908 1/20 0.36
ADRA1D P25100 1/20 0.36
ADRA1A P35348 1/20 0.36
ADRA1B P35368 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11130696 0.79 ALDH1A1 (0.49) ALDH1A1CYP3A4KMT2APABPC1APOBEC3A
SCHEMBL1202828 0.78 ALDH1A1 (0.58) ALDH1A1CYP3A4KMT2APABPC1APOBEC3A
Bromide SCHEMBL10735522 0.77 ALDH1A1 (0.47) ALDH1A1CYP3A4KMT2APABPC1APOBEC3A
SCHEMBL6378754 0.76 SMN1; SMN2 (0.43) ALDH1A1KMT2APOLBCTSAMAPK1
SCHEMBL5187281 0.75 ROCK2 (0.37) CTSAIDO1ROCK2FFAR1KCNK3
Hydrazine SCHEMBL18138498 0.75 ALDH1A1 (0.55) ALDH1A1CYP3A4KMT2APABPC1APOBEC3A
SCHEMBL6947700 0.73 AKR1C3 (0.51) ALDH1A1CYP3A4HSD17B10MAPK1ROCK2
SCHEMBL15705106 0.72 CYP3A4 (0.52) ALDH1A1CYP3A4KMT2APOLBESR1
SCHEMBL28178916 0.72 SMN1; SMN2 (0.50) ALDH1A1CYP3A4POLBMAPK1CYP19A1
SCHEMBL29660576 0.71 ALDH1A1 (0.42) ALDH1A1CYP3A4KMT2APABPC1APOBEC3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1217001-B1 QUINUCLIDINE COMPOUNDS AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT EISAI CO LTD (JP) 2005-12-07 EP disclosed
US-6599917-B1 A squalene-synthesizing enzyme inhibitor, a cholesterol biosynthesis inhibitor and a triglyceride biosynthesis inhibitor EISAI CO., LTD. (JP) 2003-07-29 US disclosed
EP-1217001-A1 QUINUCLIDINE COMPOUNDS AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT Eisai Co., Ltd. (JP) 2002-06-26 EP disclosed