SCHEMBL6378754

SCHEMBL6378754

COc1cc(C(O)c2ccccc2)ccn1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.43
CNR2 P34972 1/20 0.43
LMNA P02545 1/20 0.41
KDM4E B2RXH2 1/20 0.41
LOX P28300 1/20 0.41
LOXL2 Q9Y4K0 1/20 0.41
BRD4 O60885 1/20 0.39
CREBBP Q92793 1/20 0.39
MAPK1 P28482 1/20 0.39
KDM4A O75164 1/20 0.38
KDM4C Q9H3R0 1/20 0.38
KMT2A Q03164 3/20 0.38
ACHE P22303 2/20 0.38
CTSA P10619 1/20 0.38
ALDH1A1 P00352 1/20 0.38
POLB P06746 1/20 0.38
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37
KDM5A P29375 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26988372 0.84 LOX (0.39) SMN1; SMN2LMNALOXLOXL2MAPK1
SCHEMBL6375181 0.83 BRD4 (0.46) SMN1; SMN2CNR2LMNAKDM4EBRD4
SCHEMBL23882951 0.80 BRD4 (0.39) LOXLOXL2BRD4KMT2AACHE
SCHEMBL9366832 0.79 LOX (0.46) LOXLOXL2ACHE
SCHEMBL22585542 0.77 LOX (0.44) LOXLOXL2ACHECYP2C19KDM5A
SCHEMBL19992429 0.77 LOX (0.44) LOXLOXL2ACHECTSA
SCHEMBL10406643 0.77 SMN1; SMN2 (0.47) SMN1; SMN2LMNAKDM4EBRD4CREBBP
SCHEMBL15922040 0.77 SMN1; SMN2 (0.47) SMN1; SMN2LMNAKDM4EALDH1A1CYP1A2
SCHEMBL6375219 0.76 ALDH1A1 (0.40) MAPK1KMT2ACTSAALDH1A1POLB
SCHEMBL14065341 0.75 KMT2A (0.51) SMN1; SMN2CNR2LMNAKDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100334085-C Quinuclidine compound and medicine containing the same as active ingredient EISAI R & D CO LTD (JP) 2007-08-29 CN disclosed
EP-1217001-B1 QUINUCLIDINE COMPOUNDS AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT EISAI CO LTD (JP) 2005-12-07 EP disclosed
US-6599917-B1 A squalene-synthesizing enzyme inhibitor, a cholesterol biosynthesis inhibitor and a triglyceride biosynthesis inhibitor EISAI CO., LTD. (JP) 2003-07-29 US disclosed
CN-1377349-A Quinuclidine compound and medicine containing the same as active ingredient EISAI CO LTD (JP) 2002-10-30 CN disclosed
EP-1217001-A1 QUINUCLIDINE COMPOUNDS AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT Eisai Co., Ltd. (JP) 2002-06-26 EP disclosed