SCHEMBL6384608

SCHEMBL6384608

O=C(Oc1cc(Cl)cs1)N1CCN(c2nccc3sc(S(=O)(=O)Cc4ccc(F)c(F)c4)cc23)CC1.[LiH]

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 7/20 0.36
TRPV1 Q8NER1 3/20 0.34
AKT1 P31749 3/20 0.34
GRM4 Q14833 2/20 0.34
AKT2 P31751 1/20 0.34
AKT3 Q9Y243 1/20 0.34
IDE P14735 1/20 0.31
MALT1 Q9UDY8 1/20 0.30
P2RY12 Q9H244 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1776231 0.84 AKT1 (0.40) AKT1GRM4AKT2AKT3P2RY12
SCHEMBL1774986 0.83 GRIA1 (0.41) AKT1AKT2AKT3
SCHEMBL1776952 0.72 P2RY12 (0.41) AKT1AKT2AKT3P2RY12
SCHEMBL1776820 0.72 MEN1 (0.47)
SCHEMBL1775701 0.72 TRPV1 (0.40) TRPA1TRPV1
SCHEMBL1775123 0.72 ALDH1A1 (0.42) AKT1AKT2AKT3P2RY12
SCHEMBL1776477 0.71 AKT1 (0.40) TRPA1TRPV1AKT1AKT2AKT3
SCHEMBL1775510 0.71 ACHE (0.48)
SCHEMBL1776052 0.71 TRPA1 (0.41) TRPA1TRPV1IDE
SCHEMBL1774709 0.70 TRPA1 (0.42) TRPA1TRPV1GRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1513828-A1 NEW COMPOUNDS USEFUL FOR THE TREATMENT OF OBESITY, TYPE II DIABETES AND CNS DISORDERS Biovitrum AB (SE) 2005-03-16 EP disclosed
WO-2004000828-A1 NEW COMPOUNDS USEFUL FOR THE TREATMENT OF OBESITY, TYPE II DIABETES AND CNS DISORDERS BIOVITRUM AB (SE) 2003-12-31 WO disclosed