SCHEMBL6399162

SCHEMBL6399162

C=CCN(C)CCCCCc1ccc2c(c1)CCN2C(=O)Nc1ccc(OC)cc1OC

nearest known ligand 0.53

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.53
MAPT P10636 4/20 0.53
TP53 P04637 2/20 0.46
TAS1R3 Q7RTX0 1/20 0.44
TAS1R1 Q7RTX1 1/20 0.44
TAS1R2 Q8TE23 1/20 0.44
NPSR1 Q6W5P4 1/20 0.41
LSS P48449 1/20 0.41
NOTUM Q6P988 1/20 0.40
KMT2A Q03164 3/20 0.40
MEN1 O00255 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6401002 0.89 LSS (0.49) LMNAMAPTTP53TAS1R3TAS1R1
SCHEMBL6400584 0.88 MAPT (0.51) LMNAMAPTTP53NOTUMKMT2A
SCHEMBL6403158 0.84 LSS (0.40) LMNAMAPTTP53TAS1R3TAS1R1
SCHEMBL6402854 0.84 LSS (0.48) LMNAMAPTTP53TAS1R3TAS1R1
SCHEMBL5637812 0.82 KDM4E (0.41) LMNAMAPTTP53
SCHEMBL5638204 0.81 TP53 (0.49) LMNAMAPTTP53KMT2AMEN1
SCHEMBL6404170 0.81 LSS (0.43) LMNAMAPTTP53LSSNOTUM
SCHEMBL6400266 0.81 MAPT (0.46) LMNAMAPTTP53LSSKMT2A
SCHEMBL6404049 0.80 RAB9A (0.40) LMNAMAPTTP53LSSKMT2A
SCHEMBL5637681 0.80 LSS (0.40) MAPTTP53LSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050187390-A1 Bicyclic heteroaryl derivatives GENELABS TECHNOLOGIES, INC. 2005-08-25 US disclosed
US-20050020624-A1 Dihydroindole and tetrahydroquinoline derivatives AEBI JOHANNES (CH) 2005-01-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050020624-A1 Dihydroindole and tetrahydroquinoline derivatives CYP46A1, LSS, CYP51A1 LMNA 3715/4885MAPT 3562/4885TP53 488/4885
US-20050187390-A1 Bicyclic heteroaryl derivatives HAVCR2, MAVS, ZC3HAV1 LMNA 1546/4885MAPT 2748/4885TP53 2428/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.