SCHEMBL6399894

SCHEMBL6399894

C=CCN1C(=O)c2ccccc2C1=S

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 1/20 0.69
ALDH1A1 P00352 6/20 0.49
POLB P06746 3/20 0.49
RXFP1 Q9HBX9 1/20 0.49
NPSR1 Q6W5P4 1/20 0.47
CA12 O43570 2/20 0.46
CA9 Q16790 2/20 0.46
CA2 P00918 1/20 0.46
LMNA P02545 1/20 0.46
MAPT P10636 1/20 0.46
PKM P14618 1/20 0.46
KMT2A Q03164 3/20 0.45
NPC1 O15118 1/20 0.45
TP53 P04637 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C19 P33261 1/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
MEN1 O00255 2/20 0.43
CRHBP P24387 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31377051 0.88 CASP3 (0.85) CASP3ALDH1A1POLBRXFP1NPSR1
SCHEMBL170913 0.88 CASP3 (0.85) CASP3ALDH1A1POLBRXFP1NPSR1
Methane SCHEMBL4623788 0.86 CASP3 (0.82) CASP3ALDH1A1POLBRXFP1NPSR1
SCHEMBL13442855 0.81 CASP3 (1.00) CASP3ALDH1A1POLBRXFP1NPSR1
SCHEMBL11843816 0.80 CA12 (0.48) CASP3ALDH1A1CA12CA9PKM
SCHEMBL11845945 0.80 GLS (0.53) CASP3ALDH1A1NPSR1CA12CA9
SCHEMBL11848701 0.77 TDP1 (0.51) MAPTKMT2ACYP2C19RAB9ASMN1; SMN2
SCHEMBL2359299 0.77 CASP3 (0.46) CASP3ALDH1A1CA12CA9CA2
SCHEMBL11840055 0.77 TDP1 (0.56) MAPTCYP2C19RAB9ASMN1; SMN2TDP1
SCHEMBL11445227 0.77 CYP1B1 (0.52) ALDH1A1CA12CA9LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-57042743-A None JP disclosed
JP-57042744-A None JP disclosed
US-6946458-B2 N-thiolated beta-lactams: novel antibacterial agents for methicillin-resistant Staphylococcus aureus UNIVERSITY OF SOUTH FLORIDA (US) 2005-09-20 US disclosed
US-20030191108-A1 N-thiolated beta-lactams: novel antibacterial agents for methicillin-resistant staphylococcus aureus SOUTH FLORIDA, UNIVERSITY OF 2003-10-09 US disclosed
US-4427439-A Composition for plant growth regulation GAF CORPORATION (US) 1984-01-24 US disclosed
JP-S5742744-A RUBBER COMPOSITION YOKOHAMA RUBBER CO LTD:THE 1982-03-10 JP disclosed
JP-S5742743-A RUBBER COMPOSITION YOKOHAMA RUBBER CO LTD:THE 1982-03-10 JP disclosed
JP-S05742743-A 0001-01-01 JP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030191108-A1 N-thiolated beta-lactams: novel antibacterial agents for methicillin-resistant staphylococcus aureus AAAS, TST, NRDC CASP3 1725/4885ALDH1A1 2378/4885POLB 2073/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.