SCHEMBL6400951

SCHEMBL6400951

CC(C)(C)[Si](C)(C)OC1CCCCCC(c2ccccc2)CCC1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SLC18A3 Q16572 3/20 0.40
CYP11B2 P19099 1/20 0.38
S1PR1 P21453 3/20 0.36
S1PR5 Q9H228 1/20 0.35
LIPE Q05469 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
CYP2D6 P10635 2/20 0.35
TRPA1 O75762 1/20 0.35
KMO O15229 1/20 0.35
CYP2C19 P33261 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
TSHR P16473 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6400953 0.97 SLC18A3 (0.38) SLC18A3CYP11B2LIPESIGMAR1CYP2D6
SCHEMBL6552564 0.79 PPM1D (0.34)
SCHEMBL29789152 0.77 PPM1D (0.38)
SCHEMBL7335164 0.77 PPM1D (0.35)
SCHEMBL10632475 0.75 CYP19A1 (0.37) CYP2D6CYP2C19
Methyl Alcohol SCHEMBL29180934 0.75 PPM1D (0.35)
SCHEMBL6400954 0.75 TACR1 (0.42) S1PR1CYP2C19
SCHEMBL5975213 0.74 CYP19A1 (0.31)
SCHEMBL5975217 0.74 CYP19A1 (0.31)
SCHEMBL6399788 0.73 OPRM1 (0.39) TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6949585-B2 Cyclooctanone derivatives and cyclodecanone derivative, and use thereof EISAI CO., LTD. (JP) 2005-09-27 US disclosed
US-20040082805-A1 Cyclooctanone derivatives and cyclodecanone derivative, and use thereof EISAI R&D MANAGEMENT CO., LTD. (JP) 2004-04-29 US disclosed
EP-1375465-A9 CYCLOOCTANONE DERIVATIVE AND CYCLODECANONE DERIVATIVE, AND USE THEREOF Eisai Co., Ltd. (JP) 2004-04-14 EP disclosed
EP-1375479-A1 PYRROLIDINE DERIVATIVE AND PROCESS FOR PRODUCING THE SAME Eisai Co., Ltd. (JP) 2004-01-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040082805-A1 Cyclooctanone derivatives and cyclodecanone derivative, and use thereof CCR1, CCL2, CCR5 SLC18A3 4816/4885CYP11B2 51/4885S1PR1 603/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.