SCHEMBL640651

SCHEMBL640651

CC(C)(C)C(C(=O)O)n1c(=O)[nH]c2ccccc21

nearest known ligand 0.59

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.59
B3GNT2 Q9NY97 3/20 0.49
DAO P14920 1/20 0.47
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44
MEN1 O00255 1/20 0.44
CYP1A2 P05177 1/20 0.44
KMT2A Q03164 1/20 0.44
MDM2 Q00987 1/20 0.44
GRIA1 P42261 2/20 0.41
GRIA2 P42262 2/20 0.41
GRIA3 P42263 2/20 0.41
GRIA4 P48058 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL640633 0.80 B3GNT2 (0.54) B3GNT2DAOMDM2
SCHEMBL14827575 0.79 POLB (0.59) POLBB3GNT2DAOALDH1A1HPGD
SCHEMBL27801894 0.79 POLB (0.59) POLBB3GNT2DAOALDH1A1MEN1
SCHEMBL27143489 0.78 POLB (0.58) POLBB3GNT2DAOALDH1A1HPGD
SCHEMBL14664128 0.77 POLB (0.54) POLBB3GNT2DAOALDH1A1HPGD
SCHEMBL639518 0.77 POLB (0.57) POLBDAOALDH1A1MEN1CYP1A2
SCHEMBL10833903 0.76 POLB (0.70) POLBB3GNT2DAOALDH1A1HPGD
SCHEMBL904825 0.76 POLB (0.74) POLBB3GNT2DAOALDH1A1HPGD
SCHEMBL261055 0.75 FBP1 (0.41) B3GNT2ALDH1A1
SCHEMBL261054 0.75 FBP1 (0.41) B3GNT2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8119676-B2 Substituted benzimidazolone derivatives, medicaments comprising them and their use Abbott GmbH & Co. HG (DE) 2012-02-21 US disclosed
US-8003792-B2 CGRP (Calcitonin Gene-Related Peptide); migraine and cluster headaches; 2-(5-Bromo-1'1'-dioxido-2-oxo-2',3',5',6'-tetrahydrospiro[indole-3,4'-thiopyran]-1 (2H)-yl)-N-(2'-oxo-1,1',2',3-tetrahydrospiro[indene-2,3'-pyrrolo[2,3-b]pyridin]-5-yl)acetamide for example; use with other drugs MERCK SHARP & DOHME CORP. (US) 2011-08-23 US disclosed