SCHEMBL6409547

SCHEMBL6409547

COc1ccc(-c2cc3c(Cl)ncnc3o2)cc1

nearest known ligand 0.71

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EGFR P00533 9/20 0.57
GSK3B P49841 8/20 0.57
KDR P35968 4/20 0.55
MEN1 O00255 1/20 0.51
HPGD P15428 1/20 0.51
KMT2A Q03164 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6409156 0.83 HPGD (0.57) EGFRGSK3BKDRMEN1HPGD
Gw642138X SCHEMBL5404724 0.83 EGFR (0.57) EGFRGSK3BKDR
SCHEMBL20742179 0.81 GSK3B (0.52) EGFRGSK3BKDRMEN1HPGD
SCHEMBL759984 0.80 HPGD (0.60) EGFRGSK3BKDRMEN1HPGD
SCHEMBL5450817 0.78 GSK3B (0.60) EGFRGSK3BKDR
SCHEMBL5354432 0.75 MEN1 (0.45) GSK3BKDRMEN1HPGDKMT2A
SCHEMBL6408608 0.75 KDR (0.71) EGFRGSK3BKDR
SCHEMBL5391001 0.73 GSK3B (1.00) EGFRGSK3BKDR
SCHEMBL8293366 0.71 GSK3B (1.00) GSK3BKDR
SCHEMBL9046890 0.71 ALDH1A1 (0.56) KDRMEN1HPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015000959-A1 4-AMINO-6-ARYL[2,3-D]PYRIMIDINES FOR THE INHIBITION OF EGFR TYROSINE KINASE NORWEGIAN UNIVERSITY OF SCIENCE AND TECHNOLOGY (NTNU) (NO) 2015-01-08 WO disclosed
WO-2005092896-A1 COMPOUND FOR INHIBITING TYROSINE KINASE ACTIVITY OF DDR2 PROTEIN KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2005-10-06 WO disclosed