SCHEMBL6409563

SCHEMBL6409563

O=C(NC(=S)N1CCC(=O)C(C(c2ccccc2)c2ccccc2)C1)c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.50
ALOX5 P09917 1/20 0.50
LMNA P02545 4/20 0.47
RAB9A P51151 2/20 0.47
NPC1 O15118 1/20 0.47
TACR1 P25103 2/20 0.46
GAA P10253 1/20 0.45
POLB P06746 1/20 0.45
KMT2A Q03164 3/20 0.44
MEN1 O00255 2/20 0.44
MAPT P10636 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.43
GPR6 P46095 1/20 0.43
HTT P42858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6410627 0.78 TACR1 (0.53) TACR1
SCHEMBL4487177 0.77 TACR1 (0.55) ALDH1A1TACR1KMT2A
SCHEMBL6410854 0.77 TACR1 (0.55) TACR1
SCHEMBL6405890 0.74 KMT2A (0.58) ALDH1A1LMNATACR1GAAPOLB
SCHEMBL3435702 0.74 ALDH1A1 (0.59) ALDH1A1ALOX5RAB9ANPC1GAA
SCHEMBL2079194 0.74 ALDH1A1 (0.59) ALDH1A1ALOX5RAB9ANPC1GAA
SCHEMBL2153249 0.72 TDP1 (0.67) ALDH1A1ALOX5LMNAGAAPOLB
SCHEMBL30865951 0.72 ALOX5 (0.72) ALDH1A1ALOX5GAAPOLBKMT2A
SCHEMBL19995957 0.71 NPC1 (0.56) ALDH1A1ALOX5LMNARAB9ANPC1
SCHEMBL20006108 0.71 NPC1 (0.56) ALDH1A1ALOX5LMNARAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050038072-A1 Nitrogeneous cyclic ketone derivative, process for producing the same, and use TAKEDA CHEMICAL INDUSTRIES, LTD. 2005-02-17 US disclosed
EP-1460062-A1 NITROGENOUS CYCLIC KETONE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, AND USE Takeda Chemical Industries, Ltd. (JP) 2004-09-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050038072-A1 Nitrogeneous cyclic ketone derivative, process for producing the same, and use BDKRB1, BDKRB2, TACR1 ALDH1A1 1984/4885ALOX5 2580/4885LMNA 4687/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.