SCHEMBL6412083

SCHEMBL6412083

CS(=O)(=O)Oc1ccc2cccc(N3CCN(CCc4cnc(Cc5ccc(Br)c(F)c5)[nH]4)CC3=O)c2c1

nearest known ligand 0.32

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 14/20 0.32
DRD2 P14416 9/20 0.32
HTR2A P28223 9/20 0.32
KCNH2 Q12809 5/20 0.32
SLC6A4 P31645 4/20 0.32
ADRB2 P07550 2/20 0.32
ADRB1 P08588 2/20 0.32
ADRA2A P08913 2/20 0.32
ADRA2B P18089 2/20 0.32
ADRA2C P18825 2/20 0.32
DRD1 P21728 2/20 0.32
DRD4 P21917 2/20 0.32
SLC6A2 P23975 2/20 0.32
HRH2 P25021 2/20 0.32
ADRA1D P25100 2/20 0.32
HTR2C P28335 2/20 0.32
HTR7 P34969 2/20 0.32
ADRA1A P35348 2/20 0.32
HRH1 P35367 2/20 0.32
ADRA1B P35368 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8009019 0.90 GPR52 (0.35) HTR1ADRD2HTR2AKCNH2MCHR1
SCHEMBL6412080 0.83 FNTA (0.44) FNTAPGGT1B
SCHEMBL6430353 0.73 FNTA (0.48) FNTAPGGT1B
SCHEMBL6412396 0.70 SIRT2 (0.33) HTR1ADRD2HTR2AKCNH2SLC6A4
SCHEMBL7247790 0.66 HTR5A (0.38) HTR1ADRD2HTR2AKCNH2HTR2C
Hydrochloric Acid SCHEMBL7247789 0.66 HTR5A (0.38) HTR1ADRD2HTR2AKCNH2HTR7
SCHEMBL6417857 0.62 HTR2A (0.42) HTR1ADRD2HTR2AKCNH2SLC6A4
Hydrochloric Acid SCHEMBL8175209 0.61 FNTA (0.58) FNTAPGGT1B
SCHEMBL7715094 0.60 PSEN1 (0.33)
SCHEMBL3519558 0.56 FNTA (0.58) FNTAPGGT1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1090012-A4 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO INC (US) 2005-04-06 EP disclosed
EP-1090012-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 2001-04-11 EP disclosed
WO-2000001702-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 2000-01-13 WO disclosed