SCHEMBL8009019

SCHEMBL8009019

CS(=O)(=O)Oc1ccc2cccc(N3CCN(CCc4cnc(Cc5ccc(C#N)c(F)c5)[nH]4)CC3=O)c2c1

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GPR52 Q9Y2T5 1/20 0.35
KCNH2 Q12809 5/20 0.35
KCNJ1 P48048 3/20 0.35
HTR1A P08908 5/20 0.34
HTR1D P28221 1/20 0.34
HTR1B P28222 1/20 0.34
FNTA P49354 8/20 0.34
FNTB P49356 7/20 0.34
PGGT1B P53609 5/20 0.33
DNAJA1 P31689 1/20 0.33
DRD2 P14416 4/20 0.32
HTR2A P28223 4/20 0.32
MCHR1 Q99705 2/20 0.32
DAO P14920 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6412083 0.90 HTR1A (0.32) KCNH2HTR1AHTR1DHTR1BFNTA
SCHEMBL6430353 0.84 FNTA (0.48) FNTAFNTBPGGT1B
SCHEMBL6412080 0.73 FNTA (0.44) FNTAFNTBPGGT1B
SCHEMBL7168685 0.72 FNTA (0.47) HTR1AHTR1DHTR1BFNTAFNTB
SCHEMBL7163140 0.71 FNTA (0.46) HTR1AHTR1DHTR1BFNTAFNTB
SCHEMBL6409378 0.70 HTR1A (0.35) HTR1AHTR1DHTR1BFNTAFNTB
SCHEMBL6523879 0.69 FNTA (0.62) FNTAFNTBPGGT1B
SCHEMBL7168181 0.69 FNTA (0.41) GPR52FNTAFNTBPGGT1BDNAJA1
SCHEMBL7247564 0.69 P2RX7 (0.36) KCNH2HTR1AHTR1DHTR1BFNTA
SCHEMBL6412396 0.69 SIRT2 (0.33) KCNH2HTR1AHTR1DHTR1BDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000025789-A1 A METHOD OF TREATING ENDOMETRIOSIS MERCK & CO., INC. (US) 2000-05-11 WO disclosed