SCHEMBL6414059

SCHEMBL6414059

CN(Cc1cccc(Cl)c1)C(=O)/C=C1/OC(C)(C)OC1=O

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 1/20 0.47
AOC3 Q16853 4/20 0.44
PABPC1 P11940 1/20 0.43
NPC1 O15118 1/20 0.41
GAA P10253 2/20 0.39
TP53 P04637 1/20 0.39
TSHR P16473 1/20 0.38
RECQL P46063 1/20 0.38
PYCR1 P32322 1/20 0.38
ALDH1A1 P00352 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
TACR1 P25103 1/20 0.37
ATM Q13315 1/20 0.36
AMPD2 Q01433 1/20 0.36
PIN1 Q13526 1/20 0.36
TAAR1 Q96RJ0 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6414063 1.00 RIPK1 (0.47) RIPK1AOC3PABPC1NPC1GAA
SCHEMBL6076910 0.90 TACR1 (0.42) RIPK1AOC3PABPC1NPC1TP53
SCHEMBL6076905 0.90 TACR1 (0.42) RIPK1AOC3PABPC1NPC1TP53
SCHEMBL6077341 0.87 ALDH1A1 (0.46) AOC3NPC1TP53ALDH1A1
SCHEMBL6077313 0.86 USP30 (0.47) TSHRPYCR1ALDH1A1
SCHEMBL6077308 0.86 USP30 (0.47) TSHRPYCR1ALDH1A1
SCHEMBL6420129 0.85 USP30 (0.39) RIPK1AOC3ALDH1A1TACR1
SCHEMBL6420127 0.85 USP30 (0.39) RIPK1AOC3ALDH1A1TACR1
SCHEMBL6419943 0.84 RIPK1 (0.38) RIPK1ALDH1A1
SCHEMBL6419940 0.84 RIPK1 (0.38) RIPK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050043370-A1 HIV integrase inhibitors WALKER MICHAEL A (US) 2005-02-24 US disclosed
US-6803378-B2 FOR THERAPY AND PROPHYLAXIS OF ACQUIRED IMMUNE DEFICIENCY SYNDROME (AIDS), OR ARC BRISTOL-MYERS SQUIBB COMPANY 2004-10-12 US disclosed
US-20030181490-A1 HIV integrase inhibitors WALKER MICHAEL A (US) 2003-09-25 US disclosed
US-20030027847-A1 HIV integrase inhibitors BRISTOL-MYERS SQUIBB COMPANY 2003-02-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050043370-A1 HIV integrase inhibitors AKR1C3, CBR3, CBR1 RIPK1 3528/4885AOC3 66/4885PABPC1 3796/4885
US-20030181490-A1 HIV integrase inhibitors CBR1, CCR5, CCR1 RIPK1 3530/4885AOC3 124/4885PABPC1 2285/4885
US-20030027847-A1 HIV integrase inhibitors CBR1, CCR5, CCR1 RIPK1 3530/4885AOC3 124/4885PABPC1 2285/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.