SCHEMBL6414787

SCHEMBL6414787

CCOC(=O)c1cnc2c(c(C)nn2-c2ccccc2)c1N(Cc1ccccc1)S(=O)(=O)c1ccc(F)cc1

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 5/20 0.59
MMP13 P45452 5/20 0.59
MMP9 P14780 4/20 0.59
ADAM17 P78536 4/20 0.59
NR3C1 P04150 8/20 0.47
LMNA P02545 3/20 0.43
POLB P06746 2/20 0.43
PKM P14618 1/20 0.43
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
ATM Q13315 1/20 0.42
KDM4E B2RXH2 1/20 0.42
USP2 O75604 1/20 0.42
ALDH1A1 P00352 1/20 0.42
TSHR P16473 1/20 0.42
HSD17B10 Q99714 1/20 0.42
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6290612 0.91 MMP1 (0.71) MMP1MMP13MMP9ADAM17NR3C1
SCHEMBL6290776 0.91 MMP1 (0.56) MMP1MMP13MMP9ADAM17NR3C1
SCHEMBL7151568 0.91 MMP1 (0.61) MMP1MMP13MMP9ADAM17NR3C1
SCHEMBL6293913 0.89 MMP1 (0.56) MMP1MMP13MMP9ADAM17NR3C1
SCHEMBL6289426 0.87 MMP1 (0.58) MMP1MMP13MMP9ADAM17NR3C1
SCHEMBL6293288 0.85 MMP9 (0.81) MMP1MMP13MMP9ADAM17
SCHEMBL6293214 0.84 MMP1 (0.47) MMP1MMP13MMP9ADAM17NR3C1
SCHEMBL6290764 0.82 MMP1 (0.75) MMP1MMP13MMP9ADAM17NR3C1
SCHEMBL6290784 0.82 MMP1 (0.68) MMP1MMP13MMP9ADAM17LMNA
SCHEMBL6293912 0.80 NR3C1 (0.50) MMP1MMP13MMP9ADAM17NR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6946473-B2 Preparation and use of acetylenic ortho-sulfonamido and phosphinic acid amido bicyclic heteroaryl hydroxamic acids as TACE inhibitors WYETH HOLDINGS CORPORATION (US) 2005-09-20 US disclosed