SCHEMBL6421735

SCHEMBL6421735

CC(C)(C)OC(=O)N1CCC(c2noc3ccc(C(F)(F)F)cc23)CC1.FC(F)(F)c1ccc2onc(C3CCNCC3)c2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1F P30939 2/20 0.44
HTR1A P08908 1/20 0.44
P2RY14 Q15391 1/20 0.43
GPR119 Q8TDV5 3/20 0.42
HDAC4 P56524 2/20 0.42
HTT P42858 1/20 0.42
MAPT P10636 2/20 0.41
KDM4E B2RXH2 1/20 0.41
THRB P10828 1/20 0.41
JAK2 O60674 2/20 0.41
JAK3 P52333 2/20 0.41
JAK1 P23458 1/20 0.41
TYK2 P29597 1/20 0.41
STS P08842 1/20 0.41
PTK2 Q05397 1/20 0.40
TGFBR1 P36897 1/20 0.40
ALDH1A1 P00352 1/20 0.40
GAA P10253 1/20 0.40
HPGD P15428 1/20 0.40
TSHR P16473 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2959207 0.94 HTR1F (0.48) HTR1FHTR1AP2RY14GPR119HDAC4
SCHEMBL2955792 0.82 HTR2C (0.48) HTR1FHTR1A
SCHEMBL17495424 0.81 GPR119 (0.45) HTR1FHTR1AGPR119HTTMAPT
SCHEMBL17495459 0.81 GPR119 (0.45) HTR1FHTR1AGPR119HTTMAPT
SCHEMBL2955169 0.77 DRD2 (0.57)
SCHEMBL21679583 0.76 HTR2A (0.52) HTR1AGPR119MAPTKDM4ETHRB
SCHEMBL17495534 0.74 MEN1 (0.44) HTR1FHTR1AGPR119HTTKDM4E
SCHEMBL2962549 0.73 GPR119 (0.46) GPR119HDAC4MAPTKDM4ETHRB
SCHEMBL13201170 0.73 HTR2C (0.48)
SCHEMBL1093627 0.73 STS (0.50) P2RY14GPR119MAPTKDM4ETHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1362039-B1 HETEROCYCLIC SUBSTITUTED CARBONYL DERIVATIVES AND THEIR USE AS DOPAMINE D3 RECEPTOR LIGANDS AVENTIS PHARMA INC (US) 2005-12-21 EP disclosed