SCHEMBL6423359

SCHEMBL6423359

O=C1N(Cc2ccccc2-c2ccco2)CCCC12CCNCC2

nearest known ligand 0.64

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 16/20 0.64
HCRTR1 O43613 12/20 0.64
OPRM1 P35372 3/20 0.43
OPRD1 P41143 3/20 0.43
MAPT P10636 2/20 0.43
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
ALDH1A1 P00352 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2130959 0.80 HCRTR2 (0.71) HCRTR2HCRTR1
SCHEMBL2026883 0.78 HCRTR2 (1.00) HCRTR2HCRTR1
SCHEMBL6430669 0.76 HCRTR2 (0.73) HCRTR2HCRTR1
SCHEMBL12641223 0.76 HCRTR2 (0.63) HCRTR2HCRTR1
SCHEMBL6422976 0.76 HCRTR2 (0.44) HCRTR2HCRTR1
Hydrochloric Acid SCHEMBL2022807 0.75 HCRTR2 (0.62) HCRTR2HCRTR1
SCHEMBL12641233 0.75 MEN1 (0.64) HCRTR2HCRTR1MEN1KMT2AALDH1A1
SCHEMBL2026638 0.73 HCRTR2 (0.63) HCRTR2HCRTR1
SCHEMBL32667418 0.73 LMNA (0.51) HCRTR2HCRTR1OPRM1OPRD1MAPT
SCHEMBL2025002 0.72 HCRTR2 (0.70) HCRTR2HCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012055888-A1 DIAZA-SPIRO[5.5]UNDECANES USEFUL AS OREXIN RECEPTOR ANTAGONISTS NOVARTIS AG (CH) 2012-05-03 WO disclosed