SCHEMBL6423549

SCHEMBL6423549

CN(C)C(CC=O)c1cc(F)ccc1F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.37
CES1 P23141 2/20 0.37
PSEN1 P49768 6/20 0.37
PSEN2 P49810 6/20 0.37
APH1B Q8WW43 6/20 0.37
NCSTN Q92542 6/20 0.37
APH1A Q96BI3 6/20 0.37
PSENEN Q9NZ42 6/20 0.37
RIPK1 Q13546 1/20 0.33
DPP4 P27487 2/20 0.32
DPP9 Q86TI2 2/20 0.32
ACKR3 P25106 1/20 0.31
HTT P42858 1/20 0.31
OPRM1 P35372 3/20 0.31
MEN1 O00255 1/20 0.31
MAPT P10636 1/20 0.31
HPGD P15428 1/20 0.31
KMT2A Q03164 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
OPRL1 P41146 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4432794 0.87 CES2 (0.37) CES2CES1RIPK1ACKR3HTT
SCHEMBL4425980 0.76 AOC3 (0.40) HTTOPRM1KMT2AL3MBTL1
SCHEMBL4435860 0.75 CES2 (0.36) CES2CES1OPRM1MAPTOPRL1
SCHEMBL3829073 0.74 OPRM1 (0.47) OPRM1OPRL1
SCHEMBL4429231 0.74 CES2 (0.41) CES2CES1RIPK1OPRM1
SCHEMBL4593455 0.74 CES2 (0.41) CES2CES1PSEN1PSEN2APH1B
SCHEMBL6421263 0.73 CES2 (0.32) CES2CES1OPRM1OPRL1
SCHEMBL20640522 0.67 APLNR (0.39) CES2CES1PSEN1PSEN2APH1B
SCHEMBL31257263 0.67 APLNR (0.39) CES2CES1PSEN1PSEN2APH1B
SCHEMBL19801164 0.67 NISCH (0.38) HTTOPRM1MEN1HPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1527050-A1 QUINOLINE DERIVATIVES AND THEIR USE AS MYCOBACTERIAL INHIBITORS JANSSEN PHARMACEUTICA N.V. (BE) 2005-05-04 EP disclosed
WO-2004011436-A1 QUINOLINE DERIVATIVES AND THEIR USE AS MYCOBACTERIAL INHIBITORS JANSSEN PHARMACEUTICA N.V. (BE) 2004-02-05 WO disclosed