SCHEMBL642432

SCHEMBL642432

NC(=O)c1ccc(N2CCC(C(=O)O)CC2)cc1Oc1ccc(Cl)cc1Cl

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 10/20 0.48
FFAR1 O14842 2/20 0.45
L3MBTL1 Q9Y468 2/20 0.45
ALDH1A1 P00352 1/20 0.45
POLB P06746 1/20 0.45
GAA P10253 1/20 0.45
HPGD P15428 1/20 0.45
AKR1C3 P42330 1/20 0.45
EPHX2 P34913 1/20 0.40
F10 P00742 1/20 0.40
MAPT P10636 1/20 0.39
TTR P02766 1/20 0.39
SCN9A Q15858 1/20 0.39
CSF1R P07333 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL641984 0.87 NOTUM (0.50) NOTUMFFAR1AKR1C3MAPTSCN9A
SCHEMBL642235 0.85 NOTUM (0.48) NOTUMFFAR1ALDH1A1GAAAKR1C3
SCHEMBL640945 0.76 NOTUM (0.53) NOTUMPOLBSCN9A
SCHEMBL641081 0.76 FFAR4 (0.55) NOTUMSCN9A
SCHEMBL2557442 0.75 NOTUM (0.59) NOTUMFFAR1L3MBTL1POLBAKR1C3
Cyclopropane Carboxylic Acid SCHEMBL28423298 0.73 SMN1; SMN2 (0.53) NOTUML3MBTL1ALDH1A1GAAHPGD
SCHEMBL12716971 0.72 NEK2 (0.54) NOTUM
SCHEMBL3215648 0.72 NOTUM (0.59) NOTUMAKR1C3
SCHEMBL30755065 0.72 NOTUM (0.59) NOTUMAKR1C3
SCHEMBL2073478 0.72 NOTUM (0.81) NOTUMFFAR1ALDH1A1POLBHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8119627-B2 Heterocyclic compounds as inhibitors of 17beta-HSD3 STERIX LIMITED (GB) 2012-02-21 US disclosed