SCHEMBL642235

SCHEMBL642235

NC(=O)c1ccc(N2CCC(C(=O)O)CC2)cc1Oc1cc(Cl)cc(Cl)c1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 12/20 0.48
AKR1C3 P42330 1/20 0.44
SCN9A Q15858 2/20 0.42
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
GAA P10253 1/20 0.41
FFAR4 Q5NUL3 1/20 0.41
FFAR1 O14842 1/20 0.40
SYK P43405 1/20 0.39
PRSS1 P07477 1/20 0.38
PRSS2 P07478 1/20 0.38
PRSS3 P35030 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL641984 0.91 NOTUM (0.50) NOTUMAKR1C3SCN9AFFAR4FFAR1
SCHEMBL642432 0.85 NOTUM (0.48) NOTUMAKR1C3SCN9AALDH1A1GAA
SCHEMBL641081 0.82 FFAR4 (0.55) NOTUMSCN9AFFAR4
SCHEMBL640945 0.82 NOTUM (0.53) NOTUMSCN9AKDM4EFFAR4
SCHEMBL2073107 0.75 NOTUM (0.81) NOTUMAKR1C3KDM4EFFAR4FFAR1
SCHEMBL2557442 0.74 NOTUM (0.59) NOTUMAKR1C3FFAR1
SCHEMBL1817248 0.72 NOTUM (0.60) NOTUMFFAR4
SCHEMBL12716971 0.72 NEK2 (0.54) NOTUM
SCHEMBL3215648 0.71 NOTUM (0.59) NOTUMAKR1C3
SCHEMBL30755065 0.71 NOTUM (0.59) NOTUMAKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8119627-B2 Heterocyclic compounds as inhibitors of 17beta-HSD3 STERIX LIMITED (GB) 2012-02-21 US disclosed