SCHEMBL6426765

SCHEMBL6426765

C1=C(c2ccc3cc[nH]c3c2)CCN2CCC[C@@H]12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK11 Q15759 1/20 0.43
MAPK14 Q16539 1/20 0.43
BRD4 O60885 1/20 0.36
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35
MAPT P10636 2/20 0.35
HPGD P15428 2/20 0.35
HSD17B10 Q99714 2/20 0.35
MTOR P42345 2/20 0.35
PIK3CD O00329 1/20 0.35
ABL1 P00519 1/20 0.35
EGFR P00533 1/20 0.35
HCK P08631 1/20 0.35
SRC P12931 1/20 0.35
KDR P35968 1/20 0.35
PIK3CA P42336 1/20 0.35
PIK3CB P42338 1/20 0.35
PIK3CG P48736 1/20 0.35
EPHB4 P54760 1/20 0.35
PRKDC P78527 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6426242 1.00 MAPK11 (0.43) MAPK11MAPK14BRD4KDM4EALDH1A1
SCHEMBL15785424 0.75 MAPK11 (0.45) MAPK11MAPK14KDM4EALDH1A1MAPT
SCHEMBL6428639 0.73 HTR6 (0.47) BRD4KDM4EALDH1A1MAPTHPGD
SCHEMBL6428641 0.73 HTR6 (0.47) BRD4KDM4EALDH1A1MAPTHPGD
SCHEMBL7006008 0.69 HTR1D (0.62) BRD4
SCHEMBL7007905 0.69 SLC6A4 (0.59)
SCHEMBL7007906 0.69 SLC6A4 (0.59)
SCHEMBL7008669 0.69 HTR1D (0.61) L3MBTL1HTR1A
SCHEMBL7012887 0.68 HTR1B (0.61) HTR1A
SCHEMBL7012884 0.68 HTR1B (0.61) HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6897215-B1 Compounds having 5-HT6 receptor antagonist activity NPS ALLELIX CORP. (CA) 2005-05-24 US disclosed
WO-2001032660-A1 COMPOUNDS HAVING 5-HT6 RECEPTOR ANTAGONIST ACTIVITY NPS ALLELIX CORP. (US) 2001-05-10 WO disclosed