SCHEMBL6427623

SCHEMBL6427623

Cc1cc(C#Cc2ccc(C(C)C(=O)O)cc2)ccc1Cn1ccnc1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 8/20 0.44
CYP11B1 P15538 1/20 0.44
CYP11B2 P19099 1/20 0.44
CYP19A1 P11511 5/20 0.40
ABL1 P00519 1/20 0.40
ABL2 P42684 1/20 0.40
ACACB O00763 1/20 0.39
LMNA P02545 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ATM Q13315 1/20 0.38
AGTR2 P50052 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6427797 0.88 TBXAS1 (0.41) TBXAS1CYP19A1ACACBLMNASMN1; SMN2
SCHEMBL5735722 0.84 TBXAS1 (0.49) TBXAS1CYP11B1CYP11B2CYP19A1ABL1
SCHEMBL5735621 0.83 TBXAS1 (0.50) TBXAS1CYP11B1CYP11B2CYP19A1
SCHEMBL7984143 0.80 TBXAS1 (0.50) TBXAS1CYP11B1CYP11B2CYP19A1ABL1
SCHEMBL5737544 0.79 TBXAS1 (0.54) TBXAS1CYP11B1CYP11B2CYP19A1ABL1
SCHEMBL29239307 0.76 TBXAS1 (0.66) TBXAS1CYP11B1CYP11B2CYP19A1LMNA
SCHEMBL5737255 0.76 CYP11B1 (0.54) CYP11B1CYP11B2CYP19A1ATM
SCHEMBL5736555 0.74 CYP11B1 (0.57) CYP11B1CYP11B2CYP19A1ATM
SCHEMBL5735891 0.74 TBXAS1 (0.47) TBXAS1CYP11B1CYP11B2CYP19A1ACACB
SCHEMBL7711978 0.71 PTGS1 (0.36) ACACBLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6855512-B2 Methods for identifying inhibitors of cytochrome P450RAI ALLERGAN, INC. (US) 2005-02-15 US disclosed
US-6369225-B1 ENZYME INHIBITORS ALLERGAN SALES, INC. 2002-04-09 US disclosed
US-6369261-B1 CYCLOPROPYLBENZENE DERIVATIVE OF ACIDS OR ESTERS ALLERGAN SALES, INC. 2002-04-09 US disclosed
US-6303785-B1 SUBSTITUTED N-CYCLOPROPYLTETRAHYDROISOQUINOLINES ALLERGAN SALES, INC. 2001-10-16 US disclosed