SCHEMBL6427797

SCHEMBL6427797

CC(C)c1cc(C#Cc2ccc(C(C)C(=O)O)cc2)ccc1Cn1ccnc1

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 10/20 0.41
CYP19A1 P11511 4/20 0.39
ACACB O00763 1/20 0.38
LMNA P02545 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
AGTR2 P50052 1/20 0.37
S1PR1 P21453 1/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6427623 0.88 TBXAS1 (0.44) TBXAS1CYP19A1ACACBLMNASMN1; SMN2
SCHEMBL5735891 0.85 TBXAS1 (0.47) TBXAS1CYP19A1ACACBS1PR1
SCHEMBL5735862 0.81 TBXAS1 (0.46) TBXAS1CYP19A1AGTR2
SCHEMBL6427151 0.78 TBXAS1 (0.46) TBXAS1CYP19A1AGTR2
SCHEMBL6427160 0.78 PTGS2 (0.41) ACACBLMNA
SCHEMBL6427700 0.78 PTGS2 (0.41) LMNA
SCHEMBL6427149 0.77 TBXAS1 (0.45) TBXAS1CYP19A1AGTR2
Hydrochloric Acid SCHEMBL28198436 0.77 CYP11B1 (0.48) TBXAS1CYP19A1LMNAALDH1A1
SCHEMBL29239307 0.76 TBXAS1 (0.66) TBXAS1CYP19A1LMNA
SCHEMBL5735722 0.73 TBXAS1 (0.49) TBXAS1CYP19A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6855512-B2 Methods for identifying inhibitors of cytochrome P450RAI ALLERGAN, INC. (US) 2005-02-15 US disclosed
US-6369225-B1 ENZYME INHIBITORS ALLERGAN SALES, INC. 2002-04-09 US disclosed
US-6369261-B1 CYCLOPROPYLBENZENE DERIVATIVE OF ACIDS OR ESTERS ALLERGAN SALES, INC. 2002-04-09 US disclosed
US-6303785-B1 SUBSTITUTED N-CYCLOPROPYLTETRAHYDROISOQUINOLINES ALLERGAN SALES, INC. 2001-10-16 US disclosed