SCHEMBL6429460

SCHEMBL6429460

CCC(CO)Nc1c(C)cnc(Oc2c(C)cc(C#N)cc2C)c1OC

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.35
CYP2C19 P33261 3/20 0.35
KCNH2 Q12809 3/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2D6 P10635 2/20 0.35
ABCC3 O15438 1/20 0.35
ESR1 P03372 1/20 0.35
CYP1A2 P05177 1/20 0.35
PGR P06401 1/20 0.35
CHRM2 P08172 1/20 0.35
ABCB1 P08183 1/20 0.35
ADRA2A P08913 1/20 0.35
CHRM1 P11229 1/20 0.35
DRD1 P21728 1/20 0.35
PTGS1 P23219 1/20 0.35
SLC6A2 P23975 1/20 0.35
ADORA1 P30542 1/20 0.35
ABCC1 P33527 1/20 0.35
OPRM1 P35372 1/20 0.35
ABCC2 Q92887 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5844687 0.79 CRHR1 (0.52) CRHR1
SCHEMBL6429459 0.74 CRHR1 (0.37) CYP2C9CYP2C19KCNH2CYP3A4CYP2D6
SCHEMBL6428379 0.74 CRHR1 (0.42) CRHR1
SCHEMBL6393222 0.70 CRHR1 (0.44) CRHR1
SCHEMBL8344779 0.68 CRHR1 (0.47) PGRCRHR1
SCHEMBL5842978 0.66 CRHR1 (0.67) CRHR1
SCHEMBL5845899 0.66 CRHR1 (0.40) CRHR1
SCHEMBL6430253 0.65 CRHR1 (0.42) CRHR1
SCHEMBL6798181 0.65 CRHR1 (0.52) CYP2C9CYP2C19CYP3A4CYP1A2CRHR1
SCHEMBL5845264 0.65 CRHR1 (0.55) CRHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6844351-B1 Corticotropin releasing factor antagonists PFIZER INC. (US) 2005-01-18 US disclosed