SCHEMBL6429773

SCHEMBL6429773

Cn1ncc(/C=C/C(=O)Nc2ccc(CO[PH](=O)OCc3ccc(NC(=O)/C=C/c4cnn(C)c4-c4cccc(Cl)c4)cc3)cc2)c1-c1cccc(Cl)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.42
KMT2A Q03164 5/20 0.41
MEN1 O00255 4/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
USP2 O75604 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HTR2C P28335 2/20 0.40
MMP1 P03956 3/20 0.39
MMP2 P08253 3/20 0.39
MMP9 P14780 3/20 0.39
MCHR1 Q99705 1/20 0.39
CCNC P24863 7/20 0.39
CDK8 P49336 7/20 0.39
CDK19 Q9BWU1 1/20 0.39
LMNA P02545 3/20 0.39
MAPT P10636 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6429774 0.94 HTR2A (0.42) HTR2AKMT2AMEN1CYP1A2CYP3A4
SCHEMBL6429770 0.94 HTR2A (0.42) HTR2AKMT2AMEN1CYP1A2CYP3A4
SCHEMBL6438696 0.89 HTR2A (0.44) HTR2AKMT2AMEN1CYP3A4CYP2D6
SCHEMBL6429437 0.89 CCNC (0.46) KMT2AMEN1ALDH1A1CCNCCDK8
SCHEMBL4833244 0.84 KMT2A (0.44) HTR2AKMT2AMEN1CYP1A2CYP3A4
SCHEMBL4833270 0.84 KMT2A (0.44) HTR2AKMT2AMEN1CYP1A2CYP3A4
SCHEMBL6431326 0.84 HDAC1 (0.42) HTR2AKMT2AMEN1HTR2CCCNC
SCHEMBL6434501 0.84 CCNC (0.43) HTR2ACYP3A4CYP2C19HTR2CMMP1
SCHEMBL29208304 0.84 CCNC (0.43) HTR2ACYP3A4CYP2C19HTR2CMMP1
SCHEMBL4833850 0.83 KMT2A (0.42) HTR2AKMT2AMEN1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1556032-A1 AGENT FOR PREVENTING OR TREATING NEUROPATHY Takeda Pharmaceutical Company Limited (JP) 2005-07-27 EP disclosed
WO-2004039365-A1 AGENT FOR PREVENTING OR TREATING NEUROPATHY TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2004-05-13 WO disclosed