SCHEMBL6429809

SCHEMBL6429809

Nc1ccccc1C1(c2cccc(Br)n2)CCN(Cc2ccccc2)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 2/20 0.43
SIGMAR1 Q99720 10/20 0.42
ALDH1A1 P00352 4/20 0.42
CYP3A4 P08684 3/20 0.42
TSHR P16473 3/20 0.42
CYP2C19 P33261 3/20 0.42
TP53 P04637 2/20 0.42
CYP1A2 P05177 2/20 0.42
CYP2D6 P10635 2/20 0.42
CYP2C9 P11712 2/20 0.42
HSD17B10 Q99714 2/20 0.42
DRD2 P14416 1/20 0.41
NFKB1 P19838 1/20 0.41
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
MAPK1 P28482 1/20 0.41
HTR2B P41595 1/20 0.41
MTOR P42345 1/20 0.41
MEN1 O00255 4/20 0.40
KMT2A Q03164 4/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6045730 0.84 OPRL1 (0.41) OPRL1SIGMAR1ALDH1A1CYP3A4TSHR
SCHEMBL6045719 0.79 KDM4E (0.39) OPRL1SIGMAR1ALDH1A1CYP3A4TSHR
SCHEMBL6045515 0.75 NPFFR1 (0.46) OPRL1SIGMAR1ALDH1A1CYP3A4TSHR
SCHEMBL10916463 0.72 OPRL1 (0.70) OPRL1SIGMAR1ALDH1A1CYP3A4TSHR
SCHEMBL6045686 0.72 CYP3A4 (0.43) OPRL1SIGMAR1ALDH1A1CYP3A4TSHR
SCHEMBL14939327 0.71 SIGMAR1 (0.45) SIGMAR1ALDH1A1CYP3A4TSHRCYP2C19
SCHEMBL1056446 0.69 OPRL1 (0.49) OPRL1SIGMAR1ALDH1A1CYP3A4TSHR
SCHEMBL14939341 0.69 NPSR1 (0.65) SIGMAR1ALDH1A1DRD2HTR2AHTR2C
Oxalic Acid SCHEMBL6045620 0.68 CYP2D6 (0.43) SIGMAR1CYP3A4TSHRCYP2C19CYP2D6
SCHEMBL6045553 0.67 OPRL1 (0.45) OPRL1SIGMAR1ALDH1A1CYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1559428-A1 RECEPTOR REGULATOR Takeda Pharmaceutical Company Limited (JP) 2005-08-03 EP disclosed