SCHEMBL6433355

SCHEMBL6433355

COCCCCNC(=O)C(c1ccccc1)c1ccccc1

nearest known ligand 0.63

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 6/20 0.61
ALDH1A1 P00352 2/20 0.60
NPSR1 Q6W5P4 1/20 0.60
HPGD P15428 2/20 0.58
CNR2 P34972 5/20 0.58
HTT P42858 1/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
CYP3A4 P08684 1/20 0.55
CYP2D6 P10635 1/20 0.55
CYP2C19 P33261 1/20 0.55
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6434428 0.98 CNR1 (0.60) CNR1ALDH1A1NPSR1HPGDCNR2
SCHEMBL2334318 0.83 NAAA (0.72) CNR1CNR2CYP3A4CYP2D6CYP2C19
SCHEMBL1233128 0.82 CYP3A4 (0.63) CNR1ALDH1A1NPSR1CNR2HTT
SCHEMBL6434483 0.81 NAAA (0.75) CNR1ALDH1A1CNR2HTTCYP3A4
SCHEMBL2333785 0.81 NAAA (0.75) CNR1ALDH1A1CNR2HTTCYP3A4
SCHEMBL6436285 0.81 CNR1 (0.69) CNR1CNR2CYP3A4CYP2D6CYP2C19
SCHEMBL17749476 0.80 CNR1 (0.67) CNR1CNR2HTTSMN1; SMN2
SCHEMBL7603553 0.79 CNR1 (0.71) CNR1CNR2HTTSMN1; SMN2
SCHEMBL5100260 0.78 CNR1 (0.57) CNR1ALDH1A1NPSR1CNR2HTT
Hydrochloric Acid SCHEMBL5099409 0.78 CNR1 (0.65) CNR1CNR2HTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1224163-B1 USE OF CARBONYLAMINO DERIVATIVES AGAINST CNS DISORDERS HOFFMANN LA ROCHE (CH) 2005-03-30 EP disclosed
US-6548522-B1 N-substituted 2,2-diphenylacetamide or N-substituted 2-phenyl-2-pyridinylacetamide HOFFMANN-LA ROCHE INC. 2003-04-15 US disclosed
EP-1224163-A1 USE OF CARBONYLAMINO DERIVATIVES AGAINST CNS DISORDERS F. HOFFMANN-LA ROCHE AG (CH) 2002-07-24 EP disclosed
WO-2001027070-A1 USE OF CARBONYLAMINO DERIVATIVES AGAINST CNS DISORDERS F. HOFFMANN-LA ROCHE AG (CH) 2001-04-19 WO disclosed