SCHEMBL6434210

SCHEMBL6434210

CC(C)(Cc1ccc2ccccc2c1)NC=O

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.46
CYP2A6 P11509 1/20 0.46
CASR P41180 15/20 0.45
CYP2D6 P10635 1/20 0.42
SLC6A2 P23975 1/20 0.42
SLC6A4 P31645 1/20 0.42
SLC6A3 Q01959 1/20 0.42
KCNH2 Q12809 1/20 0.42
MC4R P32245 1/20 0.41
MC5R P33032 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16592141 0.80 CYP2D6 (0.60) CYP1A2CYP2A6CASRCYP2D6SLC6A2
SCHEMBL165251 0.79 LMNA (0.59) CYP1A2CYP2D6SLC6A2
SCHEMBL4609311 0.76 ACACB (0.51) CYP1A2CYP2A6CASRCYP2D6SLC6A2
SCHEMBL16589312 0.75 CASR (0.53) CASR
SCHEMBL2260409 0.75 TAAR1 (0.41) CYP2D6
SCHEMBL564639 0.75 RIPK1 (0.39) CYP2D6SLC6A2SLC6A3
SCHEMBL19341333 0.75 CYP2A6 (0.59) CYP1A2CYP2A6CASRMC4RMC5R
SCHEMBL8824562 0.73 CASR (0.46) CYP2A6CASR
Ammonia Solution, Strong SCHEMBL27962083 0.73 CYP2A6 (0.57) CYP1A2CYP2A6CASRMC4RMC5R
SCHEMBL564806 0.73 HDAC3 (0.39) SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1288203-B1 Cyclic nitrones and pharmaceutical compositions containing them AVENTIS PHARMA INC (US) 2005-04-20 EP disclosed
EP-1288203-A1 Cyclic nitrones and pharmaceutical compositions containing them Aventis Pharmaceuticals Inc. (US) 2003-03-05 EP disclosed
US-5962469-A PREVENTION OF OXIDATION TISSUE DAMAGE BY FREE RADICALS HOECHST MARION ROUSSEL INC. (US) 1999-10-05 US disclosed
EP-0863878-A1 CYCLIC NITRONES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM HOECHST MARION ROUSSEL, INC. (US) 1998-09-16 EP disclosed
WO-1997010218-A1 CYCLIC NITRONES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM HOECHST MARION ROUSSEL, INC. (US) 1997-03-20 WO disclosed