SCHEMBL6437554

SCHEMBL6437554

Brc1ccc(C2(c3ccc(Br)cc3)OCCO2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.40
TAAR1 Q96RJ0 1/20 0.36
CYP26A1 O43174 3/20 0.36
CYP26B1 Q9NR63 2/20 0.36
RXRA P19793 2/20 0.36
RXRB P28702 1/20 0.36
CNR1 P21554 1/20 0.35
PKM P14618 1/20 0.35
ALDH1A1 P00352 4/20 0.35
USP2 O75604 1/20 0.35
ANPEP P15144 1/20 0.33
MGLL Q99685 1/20 0.32
CYP3A4 P08684 2/20 0.32
KDM4E B2RXH2 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
ALOX15 P16050 2/20 0.32
MAPK1 P28482 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3565013 0.91 ALDH1A1 (0.40) CYP26A1CYP26B1RXRARXRBCNR1
SCHEMBL3562339 0.89 CNR1 (0.39) CYP2A6CNR1PKMALDH1A1MAPK1
SCHEMBL21679404 0.82 MAOA (0.38) CYP26A1CYP26B1RXRARXRBALDH1A1
SCHEMBL587682 0.76 TAAR1 (0.42) CYP2A6TAAR1ALDH1A1CYP3A4KDM4E
SCHEMBL15908233 0.75 MAOB (0.40) CYP26A1CYP26B1RXRARXRBCYP3A4
SCHEMBL1542779 0.75 PKM (0.32) PKM
SCHEMBL15874277 0.75 CHEK2 (0.43) CYP2A6CYP26A1CYP26B1RXRARXRB
SCHEMBL17378166 0.75 ALDH1A1 (0.43) CYP26A1CYP26B1RXRARXRBALDH1A1
SCHEMBL15874310 0.75 KMT2A (0.43) CYP26A1CYP26B1RXRARXRBCNR1
SCHEMBL235335 0.75 ESR2 (0.44) CYP26A1CYP26B1RXRARXRBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2943523-A2 SILYLATED POLYARYLETHERKETONE AND METHOD FOR MANUFACTURING SAME Perpetuum-Ebner GmbH & Co. Kg (DE) 2015-11-18 EP disclosed
WO-2014108420-A2 SILYLATED POLYARYLETHERKETONE AND METHOD FOR MANUFACTURING SAME PERPETUUM-EBNER GMBH & CO. KG (DE) 2014-07-17 WO disclosed
EP-1506959-A2 Derivatised molecules for mass spectrometry OXFORD GENE TECHNOLOGY IP LIMITED (GB) 2005-02-16 EP disclosed