SCHEMBL6439532

SCHEMBL6439532

CS(=O)(=O)c1ccc(-c2[nH]nc(COCCCO)c2-c2ccc(C(F)(F)F)cc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 1/20 0.41
PTGS2 P35354 12/20 0.39
EDNRB P24530 2/20 0.36
EDNRA P25101 2/20 0.36
PTGS1 P23219 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6438715 0.88 PTGS2 (0.41) PTGS2PTGS1
SCHEMBL6441366 0.88 PTGS2 (0.39) PTGDR2PTGS2
SCHEMBL6439571 0.87 PTGS2 (0.42) PTGS2EDNRBEDNRAPTGS1
SCHEMBL6439628 0.86 PTGS2 (0.45) PTGS2PTGS1
SCHEMBL3866671 0.79 PTGS2 (0.42) PTGS2PTGS1
SCHEMBL6445697 0.78 PTGDR2 (0.44) PTGDR2PTGS2PTGS1
SCHEMBL3863350 0.78 PTGS2 (0.43) PTGS2PTGS1
SCHEMBL3863226 0.77 PTGS2 (0.42) PTGS2EDNRBEDNRAPTGS1
SCHEMBL6440238 0.77 PTGS2 (0.42) PTGS2EDNRBEDNRAPTGS1
SCHEMBL6438240 0.77 PTGS2 (0.48) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1534683-A4 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2005-08-24 EP disclosed
EP-1534683-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2005-06-01 EP disclosed
WO-2004002409-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2004-01-08 WO disclosed