SCHEMBL6445697

SCHEMBL6445697

CS(=O)(=O)c1ccc(-c2[nH]nc(CCCC(=O)O)c2-c2ccc(C(F)(F)F)cc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 1/20 0.44
AKR1C3 P42330 1/20 0.41
PTGS2 P35354 9/20 0.40
TBXAS1 P24557 2/20 0.38
TBXA2R P21731 1/20 0.38
NR1H4 Q96RI1 1/20 0.37
S1PR1 P21453 1/20 0.37
S1PR3 Q99500 1/20 0.37
PTGS1 P23219 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6441382 0.84 POLB (0.36) PTGDR2NR1H4
SCHEMBL6439532 0.78 PTGDR2 (0.41) PTGDR2PTGS2PTGS1
SCHEMBL6440845 0.74 PTGS2 (0.44) PTGS2PTGS1
SCHEMBL6441366 0.74 PTGS2 (0.39) PTGDR2PTGS2
SCHEMBL6441425 0.73 PTGS2 (0.46) AKR1C3PTGS2
SCHEMBL6442807 0.73 PTGS2 (0.43) PTGDR2PTGS2PTGS1
SCHEMBL6438225 0.72 PTGS2 (0.51) PTGS2PTGS1
SCHEMBL8766048 0.70 PTGS2 (0.53) PTGS2PTGS1
SCHEMBL3864045 0.70 EPHX2 (0.61) AKR1C3PTGS2PTGS1
SCHEMBL8640384 0.70 PTGS2 (0.45) PTGDR2PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1534683-A4 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2005-08-24 EP disclosed
EP-1534683-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2005-06-01 EP disclosed
WO-2004002409-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2004-01-08 WO disclosed