SCHEMBL6440567

SCHEMBL6440567

N#Cc1c(NCc2ncc(C(F)(F)F)cc2Cl)nc(N)nc1-c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 18/20 0.46
ADORA2A P29274 17/20 0.46
ADORA2B P29275 5/20 0.45
P2RX3 P56373 1/20 0.42
P2RX2 Q9UBL9 1/20 0.42
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6444686 0.88 RAB9A (0.42) P2RX3P2RX2KMT2A
SCHEMBL5041750 0.85 ADORA2A (0.44) ADORA1ADORA2AADORA2BP2RX3P2RX2
SCHEMBL6444797 0.83 P2RX3 (0.40) ADORA1ADORA2AP2RX3P2RX2KMT2A
SCHEMBL6443503 0.81 P2RX3 (0.38) P2RX3P2RX2KMT2A
SCHEMBL6442124 0.80 P2RX3 (0.41) ADORA2AP2RX3P2RX2KMT2A
SCHEMBL6443545 0.74 ADORA1 (0.63) ADORA1ADORA2AADORA2B
SCHEMBL6446153 0.71 ADORA2A (0.38) ADORA1ADORA2AADORA2BP2RX3P2RX2
SCHEMBL6441739 0.69 ADORA1 (0.61) ADORA1ADORA2AADORA2B
SCHEMBL6444939 0.69 APP (0.53)
SCHEMBL6443028 0.68 ADORA1 (0.60) ADORA1ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1261327-B1 ADENOSINE RECEPTOR MODULATORS HOFFMANN LA ROCHE (CH) 2005-04-27 EP disclosed
EP-1261327-A2 ADENOSINE RECEPTOR MODULATORS F.HOFFMANN-LA ROCHE AG (CH) 2002-12-04 EP disclosed
WO-2001062233-A2 ADENOSINE RECEPTOR MODULATORS F. HOFFMANN LA ROCHE AG (CH) 2001-08-30 WO disclosed