SCHEMBL6441087

SCHEMBL6441087

CS(=O)(=O)c1ccc(-c2[nH]nc(C(=O)OCCCOCc3ccccc3)c2-c2ccccc2)cc1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 2/20 0.40
PTGS2 P35354 6/20 0.39
CHRM5 P08912 1/20 0.36
CHRM1 P11229 1/20 0.36
PTGS1 P23219 3/20 0.36
ALDH1A1 P00352 2/20 0.36
LMNA P02545 1/20 0.36
NAAA Q02083 1/20 0.35
MAPK8 P45983 1/20 0.35
ITGB1 P05556 1/20 0.35
ITGA4 P13612 1/20 0.35
CYP3A4 P08684 1/20 0.35
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6438782 0.77 PTGS2 (0.52) PTGS2PTGS1
SCHEMBL6441084 0.76 PTGS2 (0.39) GHSRPTGS2ALDH1A1LMNAMAPK1
SCHEMBL6441194 0.74 PTGS2 (0.46) GHSRPTGS2PTGS1
SCHEMBL6444404 0.74 PTGS2 (0.44) PTGS2PTGS1
SCHEMBL3865463 0.73 ESR2 (0.49) PTGS2PTGS1
SCHEMBL4958867 0.71 PTGS2 (0.46) PTGS2PTGS1MAPK8
SCHEMBL3867622 0.71 CA9 (0.54) PTGS2PTGS1
SCHEMBL6470454 0.71 PTGS2 (0.49) PTGS2PTGS1
SCHEMBL6441923 0.71 GHSR (0.42) GHSRPTGS2PTGS1
SCHEMBL6620051 0.70 PTGS2 (0.55) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1534683-A4 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2005-08-24 EP disclosed
EP-1534683-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2005-06-01 EP disclosed
WO-2004002409-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2004-01-08 WO disclosed