SCHEMBL4958867

SCHEMBL4958867

COC(=O)c1n[nH]c(-c2ccc(S(C)(=O)=O)cc2)c1Cc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 5/20 0.46
MAPK8 P45983 3/20 0.45
MAPK9 P45984 1/20 0.43
MAPK10 P53779 1/20 0.43
RNASEH1 O60930 1/20 0.42
AR P10275 1/20 0.42
KDM4E B2RXH2 1/20 0.41
STAT3 P40763 1/20 0.41
HIF1A Q16665 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
CDC7 O00311 1/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40
PTGS1 P23219 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4959110 0.84 PTGS2 (0.48) PTGS2PTGS1
SCHEMBL18302451 0.78 HCAR2 (0.46) SMN1; SMN2CDC7
SCHEMBL6590005 0.78 PTGS2 (0.43) PTGS2PTGS1
SCHEMBL4958540 0.77 PTGS2 (0.44) PTGS2PTGS1
SCHEMBL4957792 0.76 CCNB2 (0.41) PTGS2PTGS1
SCHEMBL6470454 0.74 PTGS2 (0.49) PTGS2PTGS1
SCHEMBL6438782 0.73 PTGS2 (0.52) PTGS2PTGS1
SCHEMBL6441183 0.71 PTGS2 (0.43) PTGS2KDM4EPTGS1
SCHEMBL3412438 0.71 MAPK8 (0.46) MAPK8MAPK9MAPK10ARKDM4E
SCHEMBL6441087 0.71 GHSR (0.40) PTGS2MAPK8PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1542972-A4 CYCLOOXYGENASE- 2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2008-01-23 EP claimed
EP-1542972-A2 CYCLOOXYGENASE- 2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2005-06-22 EP claimed
WO-2004010945-A2 CYCLOOXYGENASE- 2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2004-02-05 WO claimed
EP-1542972-A4 CYCLOOXYGENASE- 2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2008-01-23 EP disclosed
EP-1542972-A2 CYCLOOXYGENASE- 2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2005-06-22 EP disclosed
WO-2004010945-A2 CYCLOOXYGENASE- 2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2004-02-05 WO disclosed