SCHEMBL6441554

SCHEMBL6441554

COc1ccc(-n2c(-c3ccc(C(=O)NC(c4ccccc4)c4ccccc4)cc3)nc3ccccc32)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.61
CYP3A4 P08684 1/20 0.61
GAA P10253 2/20 0.54
CNR2 P34972 1/20 0.53
HDAC1 Q13547 1/20 0.52
HDAC8 Q9BY41 1/20 0.52
HDAC6 Q9UBN7 1/20 0.52
NPSR1 Q6W5P4 2/20 0.49
RAB9A P51151 1/20 0.49
HPGDS O60760 1/20 0.47
LMNA P02545 1/20 0.47
ESR1 P03372 1/20 0.46
ESR2 Q92731 1/20 0.46
MEN1 O00255 1/20 0.46
MAPT P10636 1/20 0.46
CRHBP P24387 1/20 0.46
KMT2A Q03164 1/20 0.46
CRHR2 Q13324 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
HPGD P15428 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6440445 0.91 CNR2 (0.53) ALDH1A1CYP3A4CNR2HDAC1HDAC8
SCHEMBL6440804 0.88 ESR2 (0.62) ALDH1A1CYP3A4GAAHDAC1HDAC8
SCHEMBL6439260 0.84 CNR2 (0.63) ALDH1A1CNR2HDAC1HDAC8HDAC6
SCHEMBL6441068 0.83 CNR2 (0.62) ALDH1A1CNR2HDAC1HDAC8HDAC6
SCHEMBL6470830 0.82 HPGDS (0.48) ALDH1A1CYP3A4GAAHDAC1HDAC8
SCHEMBL6912346 0.80 ALDH1A1 (0.67) ALDH1A1GAACNR2HDAC1HDAC8
SCHEMBL6439734 0.80 ESR2 (0.60) ALDH1A1CYP3A4GAACNR2NPSR1
SCHEMBL6438788 0.79 ESR2 (0.62) ALDH1A1GAACNR2HDAC1HDAC8
SCHEMBL6439028 0.79 ESR1 (0.67) ALDH1A1CYP3A4GAACNR2HDAC1
SCHEMBL30746859 0.79 ESR1 (0.67) ALDH1A1CYP3A4GAACNR2HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1517897-A2 BENZIMIDAZOLE COMPOUNDS AND THEIR USE AS ESTROGEN AGONISTS/ANTAGONISTS Pfizer Products Inc. (US) 2005-03-30 EP disclosed
WO-2004000817-A2 BENZIMIDAZOLE COMPOUNDS AND THEIR USE AS ESTROGEN AGONISTS/ANTAGONISTS PFIZER PRODUCTS INC. (US) 2003-12-31 WO disclosed