SCHEMBL6441622

SCHEMBL6441622

Cc1cc(C)cc(/C=C/C=O)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABBR2 O75899 1/20 0.48
GABBR1 Q9UBS5 1/20 0.48
ALDH1A1 P00352 4/20 0.46
TRPA1 O75762 2/20 0.46
ALOX5 P09917 2/20 0.46
LMNA P02545 1/20 0.46
MAPK1 P28482 1/20 0.46
XDH P47989 2/20 0.43
KDM4E B2RXH2 1/20 0.43
MAPT P10636 1/20 0.43
CDK4 P11802 4/20 0.42
CCND1 P24385 4/20 0.42
CCNB2 O95067 3/20 0.42
CDK1 P06493 3/20 0.42
CCNB1 P14635 3/20 0.42
CCNB3 Q8WWL7 3/20 0.42
ERN1 O75460 1/20 0.34
TSHR P16473 2/20 0.33
CYP2A6 P11509 1/20 0.33
MTNR1A P48039 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6441626 1.00 GABBR2 (0.48) GABBR2GABBR1ALDH1A1TRPA1ALOX5
SCHEMBL18255047 0.85 GABBR2 (0.42) GABBR2GABBR1ALDH1A1TRPA1ALOX5
SCHEMBL29350410 0.84 ALDH1A1 (0.40) GABBR2GABBR1ALDH1A1ALOX5TSHR
SCHEMBL19968585 0.84 ALDH1A1 (0.40) GABBR2GABBR1ALDH1A1ALOX5TSHR
SCHEMBL8011123 0.82 GABBR2 (0.51) GABBR2GABBR1ALDH1A1TRPA1ALOX5
SCHEMBL8011119 0.82 GABBR2 (0.51) GABBR2GABBR1ALDH1A1TRPA1ALOX5
SCHEMBL25870288 0.80 GABBR2 (0.42) GABBR2GABBR1ALDH1A1TRPA1ALOX5
SCHEMBL38660766 0.78 GABBR2 (0.47) GABBR2GABBR1ALDH1A1TRPA1ALOX5
SCHEMBL3692947 0.78 ALDH1A1 (0.44) ALDH1A1ALOX5TSHRTPMTPTGS1
SCHEMBL3692946 0.78 ALDH1A1 (0.44) ALDH1A1ALOX5TSHRTPMTPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1606251-A2 INHIBITORS OF THE BINDING OF CHEMOKINES I-TAC OR SDF-1 TO THE CCXCKR2 RECEPTOR ChemoCentryx Inc (US) 2005-12-21 EP disclosed
WO-2004058705-A2 INHIBITORS OF THE BINDING OF CHEMOKINES I-TAC OR SDF-1 TO THE CCXCKR2 RECEPTOR CHEMOCENTRYX (US) 2004-07-15 WO disclosed
US-3992472-A Synthesis of ethylenically unsaturated compounds from aldehydes or ketones E. I. DU PONT DE NEMOURS AND COMPANY (US) 1976-11-16 US disclosed