SCHEMBL6442258

SCHEMBL6442258

CCCCOC(=O)NCC(C(=O)NCC#N)c1ccc(O)cc1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.48
NPC1 O15118 3/20 0.48
RAB9A P51151 3/20 0.48
LMNA P02545 2/20 0.48
CTSS P25774 11/20 0.46
CTSK P43235 8/20 0.46
CTSL P07711 8/20 0.45
ESR1 P03372 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2D6 P10635 1/20 0.45
TSHR P16473 1/20 0.45
MAPK1 P28482 1/20 0.45
CYP2C19 P33261 1/20 0.45
NR1H2 P55055 1/20 0.45
RNASEL Q05823 1/20 0.45
CTSB P07858 4/20 0.44
HPGD P15428 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6442459 0.96 SMN1; SMN2 (0.54) SMN1; SMN2NPC1RAB9ALMNACTSS
SCHEMBL6443791 0.91 NPC1 (0.59) SMN1; SMN2NPC1RAB9ALMNACTSS
SCHEMBL6446503 0.90 SMN1; SMN2 (0.43) SMN1; SMN2NPC1RAB9ALMNACTSS
SCHEMBL6822170 0.88 CTSS (0.49) CTSSCTSKCTSLESR1CTSB
SCHEMBL6443769 0.86 NPC1 (0.65) SMN1; SMN2NPC1RAB9ALMNACTSS
SCHEMBL6446330 0.86 SMN1; SMN2 (0.48) SMN1; SMN2NPC1RAB9ALMNAESR1
SCHEMBL6445473 0.86 CTSS (0.49) CTSSCTSKCTSLESR1CTSB
SCHEMBL6443482 0.84 CTSS (0.44) CTSSCTSKCTSLESR1CTSB
SCHEMBL6447927 0.84 CTSK (0.52) CTSSCTSKCTSLESR1CTSB
SCHEMBL6442277 0.84 NPC1 (0.49) SMN1; SMN2NPC1RAB9ALMNACTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed