SCHEMBL6443340

SCHEMBL6443340

CCCC(CCC)C(=O)NC(CSC)C(=O)N(C#N)CC

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 4/20 0.37
HDAC7 Q8WUI4 2/20 0.37
HDAC6 Q9UBN7 2/20 0.37
HDAC9 Q9UKV0 2/20 0.37
HDAC5 Q9UQL6 2/20 0.37
HDAC3 O15379 3/20 0.36
HDAC4 P56524 3/20 0.36
HDAC1 Q13547 3/20 0.36
HDAC2 Q92769 3/20 0.36
CTSS P25774 2/20 0.33
CTSK P43235 2/20 0.33
HDAC10 Q969S8 1/20 0.31
HDAC11 Q96DB2 1/20 0.31
PDF Q9HBH1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6446658 0.85 HDAC8 (0.38) HDAC8HDAC7HDAC6HDAC9HDAC5
SCHEMBL6443391 0.82 HDAC8 (0.35) HDAC8HDAC7HDAC6HDAC9HDAC5
SCHEMBL6019408 0.81 KDM4E (0.33) CTSSCTSK
SCHEMBL6020453 0.80 CTSS (0.34) CTSSCTSK
SCHEMBL6019363 0.80 TGFBR1 (0.40)
SCHEMBL6019807 0.78 MEN1 (0.35) CTSSCTSK
SCHEMBL6442534 0.78 HDAC3 (0.62) HDAC8HDAC3HDAC4HDAC1HDAC2
SCHEMBL6445556 0.77 HDAC3 (0.49) HDAC8HDAC3HDAC4HDAC1HDAC2
SCHEMBL6020112 0.77 TSHR (0.35)
SCHEMBL6019181 0.76 EPHX1 (0.35) CTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed