SCHEMBL6443391

SCHEMBL6443391

CCCC(CCC)C(=O)NC(CS(C)(=O)=O)C(=O)N(C#N)CC

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 4/20 0.35
HDAC3 O15379 3/20 0.35
HDAC4 P56524 3/20 0.35
HDAC1 Q13547 3/20 0.35
HDAC2 Q92769 3/20 0.35
HDAC7 Q8WUI4 2/20 0.35
HDAC6 Q9UBN7 2/20 0.35
HDAC9 Q9UKV0 2/20 0.35
HDAC5 Q9UQL6 2/20 0.35
HDAC10 Q969S8 1/20 0.35
HDAC11 Q96DB2 1/20 0.35
CTSS P25774 1/20 0.32
CTSK P43235 1/20 0.32
CA1 P00915 2/20 0.32
CA2 P00918 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6446342 0.86 HDAC8 (0.36) HDAC8HDAC3HDAC4HDAC1HDAC2
SCHEMBL6020336 0.82 CTSS (0.32) CTSSCTSK
SCHEMBL6443340 0.82 HDAC8 (0.37) HDAC8HDAC3HDAC4HDAC1HDAC2
SCHEMBL6019892 0.81 CTSS (0.31) CTSSCTSK
SCHEMBL6021042 0.81 TGFBR1 (0.41)
SCHEMBL6020343 0.79 CTSL (0.33) CTSSCTSK
SCHEMBL6019375 0.78 TSHR (0.33)
SCHEMBL6021000 0.78 SMN1; SMN2 (0.33) CTSSCTSK
SCHEMBL6020501 0.77 CTSS (0.32) CTSSCTSK
SCHEMBL6019423 0.77 POLB (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed