SCHEMBL6444192

SCHEMBL6444192

N#CCCNC(=O)C(CNC(=O)c1ccccc1C(=O)O)c1csc2ccccc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.40
TAAR1 Q96RJ0 1/20 0.40
KMT2A Q03164 4/20 0.38
APEX1 P27695 1/20 0.38
CTSK P43235 3/20 0.36
CTSS P25774 2/20 0.36
CTSL P07711 1/20 0.36
POLB P06746 1/20 0.36
HPGD P15428 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
MEN1 O00255 2/20 0.35
ALOX5 P09917 1/20 0.35
CMA1 P23946 1/20 0.35
HDAC3 O15379 1/20 0.34
HDAC4 P56524 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC10 Q969S8 1/20 0.34
HDAC11 Q96DB2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6021888 0.91 CTSK (0.44) KDM4ETAAR1KMT2AAPEX1CTSK
SCHEMBL6446396 0.89 HPGD (0.37) KDM4EKMT2ACTSKCTSSCTSL
SCHEMBL6021296 0.89 CTSL (0.38) CTSKCTSSCTSLSMN1; SMN2ALOX5
SCHEMBL6443355 0.87 HPGD (0.41) KMT2AHPGDMEN1LMNAMAPT
SCHEMBL6447617 0.83 CTSK (0.37) TAAR1CTSKCTSSCTSLPOLB
SCHEMBL6442386 0.83 CTSK (0.42) CTSKCTSSCTSLPOLBSMN1; SMN2
SCHEMBL6443534 0.82 HDAC6 (0.37) CTSKCTSSCTSLSMN1; SMN2ALOX5
SCHEMBL6821937 0.81 CTSK (0.43) KDM4EKMT2ACTSKCTSSCTSL
SCHEMBL6449675 0.81 CTSK (0.39) TAAR1CTSKCTSSCTSLPOLB
SCHEMBL6448077 0.81 KDM4E (0.54) KDM4ETAAR1KMT2AAPEX1CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed