SCHEMBL6443534

SCHEMBL6443534

N#CCCNC(=O)C(CNC(=O)c1ccc(CCl)cc1)c1csc2ccccc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 3/20 0.37
HDAC1 Q13547 2/20 0.37
GCGR P47871 1/20 0.34
GPX4 P36969 1/20 0.34
CTSK P43235 2/20 0.33
CMA1 P23946 2/20 0.33
ALOX5 P09917 1/20 0.33
F9 P00740 1/20 0.33
CTSL P07711 1/20 0.33
CTSS P25774 1/20 0.33
GUSB P08236 1/20 0.33
SMN1; SMN2 Q16637 4/20 0.32
TP53 P04637 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
HDAC3 O15379 1/20 0.31
HDAC4 P56524 1/20 0.31
HDAC7 Q8WUI4 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
HDAC9 Q9UKV0 1/20 0.31
HDAC5 Q9UQL6 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6447552 0.91 CTSK (0.42) HDAC6HDAC1CTSKCTSLCTSS
SCHEMBL6021296 0.90 CTSL (0.38) HDAC6HDAC1GPX4CTSKCMA1
SCHEMBL6446480 0.90 GUSB (0.36) HDAC6GPX4CTSKCMA1ALOX5
SCHEMBL6443721 0.85 CMA1 (0.38) HDAC6CMA1F9SMN1; SMN2TP53
SCHEMBL6444192 0.82 KDM4E (0.40) HDAC6HDAC1CTSKCMA1ALOX5
SCHEMBL6446396 0.81 HPGD (0.37) HDAC6HDAC1CTSKCMA1ALOX5
SCHEMBL6442019 0.81 CTSS (0.42) CTSKCTSLCTSSGUSBSMN1; SMN2
SCHEMBL6448205 0.81 CTSL (0.47) CTSKALOX5CTSLCTSS
SCHEMBL6446814 0.81 CTSL (0.41) CTSKCTSLCTSS
SCHEMBL6442386 0.81 CTSK (0.42) CTSKCMA1ALOX5CTSLCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed