SCHEMBL6444345

SCHEMBL6444345

CSCC(NC(=O)NCCc1ccccc1)C(=O)NCCC#N

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ANPEP P15144 1/20 0.54
KMT2A Q03164 3/20 0.52
MEN1 O00255 1/20 0.51
TSHR P16473 1/20 0.51
PSMB1 P20618 1/20 0.47
PSMB5 P28074 1/20 0.47
PSMB2 P49721 1/20 0.47
CTSS P25774 2/20 0.45
CTSK P43235 2/20 0.45
POLB P06746 1/20 0.44
NPC1 O15118 1/20 0.44
MAPT P10636 1/20 0.44
RAB9A P51151 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6446714 0.92 ANPEP (0.57) ANPEPKMT2AMEN1TSHRPSMB1
SCHEMBL6021447 0.89 ANPEP (0.56) ANPEPCTSSCTSKMAPT
SCHEMBL6445458 0.88 KMT2A (0.67) ANPEPKMT2APSMB1PSMB5PSMB2
SCHEMBL6445490 0.85 ANPEP (0.51) ANPEPKMT2AMEN1TSHRPSMB1
SCHEMBL6442637 0.83 KMT2A (0.61) KMT2APSMB1PSMB5PSMB2CTSS
SCHEMBL6020261 0.82 CTSL (0.58) CTSSCTSK
SCHEMBL6021095 0.81 CASR (0.48) KMT2AMEN1PSMB1PSMB5PSMB2
SCHEMBL6446666 0.81 CTSS (0.57) ANPEPKMT2APSMB1PSMB5PSMB2
SCHEMBL6446628 0.81 KMT2A (0.70) ANPEPKMT2APSMB1PSMB5PSMB2
SCHEMBL6019819 0.81 CASR (0.45) CTSSCTSKNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed