SCHEMBL6445558

SCHEMBL6445558

CC(C)N(CCOc1ccc2sccc2c1)C(C)C

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.47
ESR1 P03372 2/20 0.45
ESR2 Q92731 2/20 0.45
MRGPRX4 Q96LA9 2/20 0.44
CHRNB2 P17787 1/20 0.43
CHRNA4 P43681 1/20 0.43
CA2 P00918 7/20 0.43
CA12 O43570 6/20 0.43
KCNH2 Q12809 1/20 0.41
MCHR1 Q99705 1/20 0.41
ACHE P22303 2/20 0.41
ADORA2A P29274 2/20 0.41
ADORA1 P30542 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6468074 0.79 KDM4E (0.50) MRGPRX4CA2CA12
SCHEMBL3800027 0.79 CA2 (0.49) LTA4HMRGPRX4CA2CA12
SCHEMBL828208 0.79 CA2 (0.49) LTA4HMRGPRX4CA2CA12
SCHEMBL3809957 0.77 SIGMAR1 (0.56) LTA4HMRGPRX4CA2CA12
Hydrochloric Acid SCHEMBL3815309 0.76 SIGMAR1 (0.55) LTA4HMRGPRX4CA2CA12
SCHEMBL2988516 0.75 MRGPRX4 (0.47) MRGPRX4CA2CA12
SCHEMBL5564792 0.75 MRGPRX4 (0.50) MRGPRX4CA2CA12
SCHEMBL3793751 0.75 CA2 (0.51) MRGPRX4CA2CA12
SCHEMBL3164463 0.75 NR5A1 (0.47) LTA4HMRGPRX4CA2CA12
SCHEMBL5566031 0.74 TBXAS1 (0.54) LTA4HESR1ESR2CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1594857-A2 N-MONOACYLATED O-PHENYLENEDIAMINES AS ANTI-CANCER AGENTS F. HOFFMANN-LA ROCHE AG (CH) 2005-11-16 EP disclosed
WO-2004069133-A2 N-MONOACYLATED O-PHENYLENEDIAMINES AS ANTI -CANCER AGENTS F. HOFFMANN-LA ROCHE AG (CH) 2004-08-19 WO disclosed