SCHEMBL6445645

SCHEMBL6445645

O=C(F)c1cc(Cl)c(Cl)c(Cl)c1Cl

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 6/20 0.48
HPGD P15428 5/20 0.48
HSD17B10 Q99714 5/20 0.48
CYP3A4 P08684 3/20 0.48
HSP90AA1 P07900 1/20 0.48
MAPK1 P28482 2/20 0.37
ALDH1A1 P00352 5/20 0.35
CASP1 P29466 2/20 0.35
TP53 P04637 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CRHBP P24387 1/20 0.35
CRHR2 Q13324 1/20 0.35
HIF1A Q16665 1/20 0.32
AKR1B1 P15121 1/20 0.32
KDM4E B2RXH2 1/20 0.31
MAPT P10636 1/20 0.31
AHR P35869 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9766142 0.79 KEAP1 (0.39) TSHRHPGDHSD17B10CYP3A4HSP90AA1
SCHEMBL1437003 0.78 CYP3A4 (0.48) TSHRHPGDHSD17B10CYP3A4HSP90AA1
SCHEMBL1315659 0.78 CYP3A4 (0.48) TSHRHPGDHSD17B10CYP3A4HSP90AA1
SCHEMBL8647557 0.76 CYP3A4 (0.46) TSHRHPGDHSD17B10CYP3A4HSP90AA1
SCHEMBL10498598 0.76 CYP3A4 (0.46) TSHRHPGDHSD17B10CYP3A4HSP90AA1
Fluoride SCHEMBL6445648 0.76 CYP3A4 (0.47) TSHRHPGDHSD17B10CYP3A4HSP90AA1
SCHEMBL11406014 0.74 CYP3A4 (0.43) TSHRHPGDHSD17B10CYP3A4HSP90AA1
SCHEMBL5591588 0.74 MEN1 (0.37) TSHRHPGDHSD17B10CYP3A4HSP90AA1
SCHEMBL20577112 0.74 CYP3A4 (0.43) TSHRHPGDHSD17B10CYP3A4HSP90AA1
SCHEMBL11704506 0.74 CYP3A4 (0.43) TSHRHPGDHSD17B10CYP3A4HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5565614-A FLUORINATION BAYER AKTIENGESELLSCHAFT (DE) 1996-10-15 US claimed
US-5362909-A Two stage fluorination BAYER AKTIENGESELLSCHAFT (DE) 1994-11-08 US claimed
EP-0164619-B1 2,4,5-TRIHALO OR 2,3,4,5-TETRAHALO BENZENE DERIVATIVES AND PROCESS FOR PRODUCING THEM BAYER AG (DE) 1988-10-12 EP claimed
CN-85101737-A Preparation 2,4,5-trihalogenated benzene and 2,3,4, the derivative method of 5-tetrahalogeno-benzene 1987-01-31 CN claimed
EP-0164619-A1 2,4,5-Trihalo or 2,3,4,5-tetrahalo benzene derivatives and process for producing them BAYER AG (DE) 1985-12-18 EP claimed
EP-1233010-B1 Method for production of organic fluorine compound NIPPON CATALYTIC CHEM IND (JP) 2005-06-15 EP disclosed
EP-0908438-B1 Process for the preparation of 2,3,4,5-tetrafluorobenzene derivatives BAYER AG (DE) 2003-11-26 EP disclosed
US-6613948-B1 Reacting the corresponding chlorobenzene or (chloro, fluoro)-benzene derivatives with potassium fluoride in solvent; distillation; tetrachloro benzotrifluoride, -benzoyl fluoride, or -benzonitrile as starting materials BAYER AG (DE) 2003-09-02 US disclosed
EP-0899256-B1 Method for production of organic fluorine compound NIPPON CATALYTIC CHEM IND (JP) 2003-08-06 EP disclosed
EP-1233010-A1 Method for production of organic fluorine compound Nippon Shokubai Co., Ltd. (JP) 2002-08-21 EP disclosed
US-6392084-B1 FLUORINATION OF AN ORGANO(BROMINE OR CHLORIDE) COMPOUND IN BENZONITRILE SOLVENT NIPPON SHOKUBAI CO., LTD. (JP) 2002-05-21 US disclosed
US-6114590-A Process for the preparation of polyhalogenated benzotrifluorides, benzotrichlorides and benzoyl chlorides and new trihalogenobenzotrichlorides and -benzoyl chlorides BAYER AKTIENGESELLSCHAFT (DE) 2000-09-05 US disclosed
US-5362909-A Two stage fluorination BAYER AKTIENGESELLSCHAFT (DE) 1994-11-08 US disclosed
EP-0607824-A2 Method for the production of multiply halogenated benzotrifluorides, benzotrichlorides and benzoyl chlorides as well as trihalobenzotrichlorides and -benzoyl chlorides BAYER AG (DE) 1994-07-27 EP disclosed
US-5200548-A Intermediates for bactericides BAYER AKTIENGESELLSCHAFT (DE) 1993-04-06 US disclosed
US-5072038-A Chemical intermediates for bactericides BAYER AKTIENGESELLSCHAFT (DE) 1991-12-10 US disclosed
CN-1013370-B Process for preparing derivatives of 2, 4, 5-trihalobenzenes and 2, 3, 4, 5-tetrahalobenzenes BAYER AG (DE) 1991-07-31 CN disclosed
EP-0164619-B1 2,4,5-TRIHALO OR 2,3,4,5-TETRAHALO BENZENE DERIVATIVES AND PROCESS FOR PRODUCING THEM BAYER AG (DE) 1988-10-12 EP disclosed
CN-85101737-A Preparation 2,4,5-trihalogenated benzene and 2,3,4, the derivative method of 5-tetrahalogeno-benzene 1987-01-31 CN disclosed
EP-0164619-A1 2,4,5-Trihalo or 2,3,4,5-tetrahalo benzene derivatives and process for producing them BAYER AG (DE) 1985-12-18 EP disclosed