SCHEMBL6445846

SCHEMBL6445846

CN(C#N)C(=O)C(Cc1ccc(O)cc1)NC(=O)c1cccs1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSL P07711 4/20 0.56
CTSS P25774 4/20 0.48
CTSB P07858 3/20 0.48
CTSK P43235 2/20 0.48
HSPA5 P11021 4/20 0.43
HSPA2 P54652 2/20 0.43
HSPA1A P0DMV8 1/20 0.43
HSPA9 P38646 1/20 0.43
RAB9A P51151 1/20 0.43
HPGD P15428 1/20 0.42
TSHR P16473 1/20 0.40
PYGL P06737 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6447088 0.91 CTSL (0.68) CTSLCTSSCTSBCTSKHSPA5
SCHEMBL6818989 0.87 CTSL (0.54) CTSLCTSSCTSBCTSKHSPA5
SCHEMBL6443368 0.85 CTSL (0.53) CTSLCTSSCTSBCTSKHSPA5
SCHEMBL6019209 0.83 CTSL (0.67) CTSLCTSSCTSBCTSKRAB9A
SCHEMBL6443712 0.83 CTSL (0.51) CTSLCTSSCTSBHSPA5HSPA2
SCHEMBL6443295 0.81 CTSB (0.53) CTSLCTSSCTSBCTSKHSPA5
SCHEMBL6019617 0.80 CTSL (0.53) CTSLCTSSCTSBCTSKRAB9A
SCHEMBL16993875 0.80 CTSL (0.57) CTSLHSPA5HSPA2HSPA1AHSPA9
SCHEMBL16993982 0.80 CTSL (0.57) CTSLHSPA5HSPA2HSPA1AHSPA9
SCHEMBL6020053 0.79 CTSL (0.50) CTSLCTSSCTSBCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed