SCHEMBL6446273

SCHEMBL6446273

CC(C)COC(=O)NCC(C(=O)NCCC#N)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CTSK P43235 12/20 0.48
CTSS P25774 11/20 0.48
CTSL P07711 10/20 0.46
CTSB P07858 4/20 0.44
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
POLB P06746 1/20 0.41
KDM4A O75164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6447090 0.91 CTSK (0.58) CTSKCTSSCTSLCTSB
SCHEMBL6448170 0.90 CTSK (0.42) CTSKCTSSCTSLCTSBALDH1A1
SCHEMBL6442434 0.88 POLB (0.45) CTSKCTSSCTSLCTSBALDH1A1
SCHEMBL6443928 0.87 CTSK (0.41) CTSKCTSSCTSLCTSBALDH1A1
SCHEMBL6447305 0.87 CTSS (0.43) CTSKCTSSCTSLCTSBLMNA
SCHEMBL6445366 0.87 CTSS (0.47) CTSKCTSSCTSLCTSBALDH1A1
SCHEMBL6443774 0.84 NPC1 (0.55) CTSKCTSSCTSLCTSBLMNA
SCHEMBL6443607 0.84 CTSS (0.38) CTSKCTSSCTSLCTSBALDH1A1
SCHEMBL6445439 0.83 CTSS (0.56) CTSKCTSSCTSLCTSBPOLB
SCHEMBL6445531 0.83 NPC1 (0.60) LMNAKDM4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed