SCHEMBL6446301

SCHEMBL6446301

CCCCOC(=O)NCC(C(=O)NCC#N)c1csc2ccccc12

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CTSS P25774 10/20 0.46
CTSL P07711 8/20 0.46
CTSK P43235 7/20 0.46
SMN1; SMN2 Q16637 4/20 0.44
NPC1 O15118 3/20 0.44
RAB9A P51151 3/20 0.44
LMNA P02545 1/20 0.44
CTSB P07858 4/20 0.41
ALDH1A1 P00352 2/20 0.38
CYP1A2 P05177 2/20 0.38
CYP2C19 P33261 2/20 0.38
NFKB1 P19838 1/20 0.38
STAT1 P42224 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
MAPT P10636 1/20 0.37
CYP2C9 P11712 1/20 0.37
ALOX5 P09917 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6446381 0.96 SMN1; SMN2 (0.49) CTSSCTSLCTSKSMN1; SMN2NPC1
SCHEMBL6448203 0.90 CTSS (0.48) CTSSCTSLCTSKLMNACTSB
SCHEMBL6449690 0.88 SMN1; SMN2 (0.45) CTSSCTSLCTSKSMN1; SMN2NPC1
SCHEMBL6446410 0.88 CTSS (0.48) CTSSCTSLCTSKCTSBALOX5
SCHEMBL6443383 0.87 CTSS (0.51) CTSSCTSLCTSKCTSBALOX5
SCHEMBL6445436 0.87 CTSS (0.44) CTSSCTSLCTSKCTSBALDH1A1
SCHEMBL6445530 0.86 CTSS (0.47) CTSSCTSLCTSKLMNACTSB
SCHEMBL6444043 0.83 CTSS (0.62) CTSSCTSLCTSKCTSB
SCHEMBL6446717 0.82 CTSK (0.40) CTSSCTSLCTSKSMN1; SMN2LMNA
SCHEMBL6442470 0.81 CTSK (0.45) CTSSCTSLCTSKCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed