SCHEMBL6449690

SCHEMBL6449690

CCCCCCOC(=O)NCC(C(=O)NCCC#N)c1csc2ccccc12

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.45
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
LMNA P02545 2/20 0.43
CTSL P07711 2/20 0.37
CTSS P25774 2/20 0.37
CTSK P43235 1/20 0.37
TSHR P16473 2/20 0.36
ACHE P22303 6/20 0.35
ALOX5 P09917 1/20 0.34
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6446381 0.92 SMN1; SMN2 (0.49) SMN1; SMN2NPC1RAB9ALMNACTSL
SCHEMBL6446717 0.89 CTSK (0.40) SMN1; SMN2LMNACTSLCTSSCTSK
SCHEMBL6446301 0.88 CTSS (0.46) SMN1; SMN2NPC1RAB9ALMNACTSL
SCHEMBL6449675 0.86 CTSK (0.39) NPC1RAB9ACTSLCTSSCTSK
SCHEMBL6442386 0.86 CTSK (0.42) SMN1; SMN2CTSLCTSSCTSKALOX5
SCHEMBL6446288 0.85 CTSK (0.39) LMNACTSLCTSSCTSKTSHR
SCHEMBL6450930 0.85 CTSS (0.36) CTSLCTSSCTSKALOX5ALDH1A1
SCHEMBL6443387 0.83 CTSS (0.52) CTSLCTSSCTSKALOX5
SCHEMBL6445531 0.82 NPC1 (0.60) SMN1; SMN2NPC1RAB9ALMNATSHR
SCHEMBL6448203 0.80 CTSS (0.48) LMNACTSLCTSSCTSKALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed