SCHEMBL6446342

SCHEMBL6446342

CCCC(CCC)C(=O)NC(CS(C)(=O)=O)C(=O)N(C)C#N

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 4/20 0.36
HDAC3 O15379 3/20 0.36
HDAC4 P56524 3/20 0.36
HDAC1 Q13547 3/20 0.36
HDAC2 Q92769 3/20 0.36
HDAC7 Q8WUI4 2/20 0.36
HDAC6 Q9UBN7 2/20 0.36
HDAC9 Q9UKV0 2/20 0.36
HDAC5 Q9UQL6 2/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC11 Q96DB2 1/20 0.36
CTSS P25774 2/20 0.32
CTSK P43235 2/20 0.32
CTSL P07711 1/20 0.32
CTSB P07858 1/20 0.32
CTSF Q9UBX1 1/20 0.32
PDF Q9HBH1 1/20 0.32
CA1 P00915 4/20 0.32
CA2 P00918 4/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6443391 0.86 HDAC8 (0.35) HDAC8HDAC3HDAC4HDAC1HDAC2
SCHEMBL6446658 0.81 HDAC8 (0.38) HDAC8HDAC3HDAC4HDAC1HDAC2
SCHEMBL6019926 0.78 TGFBR1 (0.43) CTSSCTSKCTSLCTSBCTSF
SCHEMBL6020060 0.78 CTSL (0.34) CTSSCTSKCTSLCTSBCTSF
SCHEMBL6021288 0.77 CTSL (0.36) CTSSCTSKCTSLCTSBCTSF
SCHEMBL6020269 0.76 SMN1; SMN2 (0.34) CTSSCTSKCTSLCTSB
SCHEMBL6019791 0.76 TSHR (0.35) CTSSCTSKCTSLCTSBCTSF
SCHEMBL6442695 0.75 HDAC3 (0.64) HDAC8HDAC3HDAC4HDAC1HDAC2
SCHEMBL6020545 0.75 PHF8 (0.36) CTSSCTSKCTSLCTSBCTSF
SCHEMBL6819030 0.74 HDAC3 (0.50) HDAC8HDAC3HDAC4HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed