SCHEMBL6447147

SCHEMBL6447147

C=CCCCCn1c(=O)c2cc(C(=O)OCc3ccccc3)sc2n(C)c1=O.Cn1c(=O)c2cc(C(=O)OCc3ccccc3)sc2n(C)c1=O.Cn1c(=O)n(Cc2cccnc2)c(=O)c2cc(C(=O)OCc3ccccc3)sc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.42
HIF1A Q16665 3/20 0.42
HTT P42858 1/20 0.42
GAA P10253 2/20 0.41
KDM4E B2RXH2 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
TRPA1 O75762 1/20 0.40
MAPK1 P28482 2/20 0.38
PKM P14618 2/20 0.37
NPSR1 Q6W5P4 2/20 0.37
MAPT P10636 2/20 0.37
LMNA P02545 2/20 0.37
BLM P54132 1/20 0.37
PARG Q86W56 2/20 0.37
MMP13 P45452 1/20 0.37
KMT2A Q03164 2/20 0.36
TDP1 Q9NUW8 2/20 0.36
GABRA1 P14867 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6255158 0.98 HIF1A (0.44) ALDH1A1HIF1AHTTGAAKDM4E
SCHEMBL6255943 0.89 HIF1A (0.48) ALDH1A1HIF1AHTTGAAKDM4E
SCHEMBL6257053 0.88 ALDH1A1 (0.41) ALDH1A1HTTGAAKDM4EMAPT
SCHEMBL6445993 0.86 HIF1A (0.53) ALDH1A1HIF1AHTTGAAKDM4E
SCHEMBL6472710 0.81 TRPA1 (0.49) ALDH1A1HIF1AKDM4ETRPA1MAPT
SCHEMBL6256050 0.81 TRPA1 (0.49) ALDH1A1HIF1AKDM4ETRPA1MAPT
SCHEMBL6252686 0.81 MMP13 (0.53) ALDH1A1KDM4ETRPA1PKMMAPT
SCHEMBL6533260 0.80 TRPA1 (0.47) ALDH1A1HIF1AHTTTRPA1MAPK1
SCHEMBL6470646 0.79 TRPA1 (0.40) ALDH1A1KDM4ETRPA1PKMMAPT
SCHEMBL6259076 0.79 ALDH1A1 (0.47) ALDH1A1HTTKDM4EMAPK1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1536786-A1 COMBINATION OF AN ALLOSTERIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 WITH CELECOXIB OR VALDECOXIB WARNER-LAMBERT COMPANY LLC (US) 2005-06-08 EP disclosed
WO-2004006913-A1 COMBINATION OF AN ALLOSTERIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 WITH CELECOXIB OR VALDECOXIB WARNER-LAMBERT COMPANY LLC (US) 2004-01-22 WO disclosed