SCHEMBL6447899

SCHEMBL6447899

CSC(CNC(=O)c1ccccc1)C(=O)NCC#N

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CTSL P07711 10/20 0.54
CTSS P25774 8/20 0.54
CTSB P07858 8/20 0.54
CTSK P43235 7/20 0.54
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
CTSV O60911 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6443785 0.89 CTSL (0.44) CTSLCTSSCTSBCTSKNPC1
SCHEMBL5526376 0.86 EPHX2 (0.52) CTSLCTSSCTSBCTSKNPC1
SCHEMBL6443960 0.85 CTSB (0.44) CTSLCTSSCTSBCTSKCTSV
SCHEMBL5517733 0.85 CTSL (0.51) CTSLCTSSCTSBCTSKNPC1
SCHEMBL6446809 0.85 KDM4E (0.51) CTSLCTSSCTSBCTSK
SCHEMBL6446731 0.84 CACNA1B (0.46) CTSLSMN1; SMN2
SCHEMBL6442984 0.84 CTSL (0.49) CTSLCTSSCTSBCTSKCTSV
SCHEMBL5524114 0.84 CTSL (0.56) CTSLCTSSCTSBCTSKSMN1; SMN2
SCHEMBL6824499 0.83 CTSL (0.62) CTSLNPC1
SCHEMBL6442378 0.83 GAA (0.47) CTSLCTSSCTSBCTSKNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed